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Items where Author is "Wenzler, T."

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Number of items: 29.

Article

Farahat, A. A. and Kumar, A. and Wenzler, T. and Brun, R. and Paul, A. and Guo, P. and Wilson, W. D. and Boykin, D. W.. (2023) Investigation of the effect of structure modification of furamidine on the DNA minor groove binding and antiprotozoal activity. Eur J Med Chem, 252. p. 115287.

Arafa, R. K. and Ismail, M. A. and Wenzler, T. and Brun, R. and Paul, A. and Wilson, W. D. and Alakhdar, A. A. and Boykin, D. W.. (2021) New antiparasitic flexible triaryl diamidines, their prodrugs and aza analogues: synthesis,; in vitro; and; in vivo; biological evaluation, and molecular modelling studies. European journal of medicinal chemistry, 222. p. 113625.

Nefertiti, A. S. G. and Batista, M. M. and Da Silva, P. B. and Batista, D. G. J. and Da Silva, C. F. and Peres, R. B. and Torres-Santos, E. C. and Cunha-Junior, E. F. and Holt, E. and Boykin, D. W. and Brun, R. and Wenzler, T. and Soeiro, M. N. C.. (2018) In Vitro and In Vivo Studies of the Trypanocidal Effect of Novel Quinolines. Antimicrobial Agents and Chemotherapy, 62 (2). e01936-17.

Gysin, M. and Braissant, O. and Gillingwater, K. and Brun, R. and Mäser, P. and Wenzler, T.. (2018) Isothermal microcalorimetry - a quantitative method to monitor Trypanosoma congolense growth and growth inhibition by trypanocidal drugs in real time. International journal for parasitology. Drugs and drug resistance, 8 (2). pp. 159-164.

Nefertiti, A. S. G. and Batista, M. M. and Da Silva, P. B. and Batista, D. G. J. and Da Silva, C. F. and Peres, R. B. and Torres-Santos, E. C. and Cunha-Junior, E. F. and Holt, E. and Boykin, D. W. and Brun, R. and Wenzler, T. and Soeiro, M. N. C.. (2018) The trypanocidal effect of novel quinolines: in vitro and in vivo studies. Antimicrobial agents and chemotherapy, 62 (2). e01936-17.

Waldsö, I. and Hallén, D. and Jansoon, M. and Suurkuusk, J. and Wenzler, T. and Braissant, O.. (2017) A well-plate format isothermal multi-channel microcalorimeter for monitoring the activity of living cells and tissues. Thermochimica acta, 652. pp. 141-149.

Farahat, A. A. and Kumar, A. and Say, M. and Wenzler, T. and Brun, R. and Paul, A. and Wilson, D. W. and Boykin, D. W.. (2017) Exploration of DAPI analogues : synthesis, antitrypanosomal activity, DNA binding and fluorescence properties. European journal of medicinal chemistry, 128. pp. 70-78.

Malebo, H. M. and Wenzler, T. and Cal, M. and Swaleh, S. M. and Omolo, M. O. and Hassanali, A. and Sequin, U. and Häussinger, D. and Dalsgaard, P. and Hamburger, M. and Brun, R. and Ndiege, I. O.. (2013) Anti-protozoal activity of aporphine and protoberberine alkaloids from Annickia kummeriae (Engl. & Diels) Setten & Maas (Annonaceae). BMC complementary and alternative medicine, Vol. 13 , 48.

Mäser, P. and Wittlin, S. and Rottmann, M. and Wenzler, T. and Kaiser, M. and Brun, R.. (2012) Antiparasitic agents : new drugs on the horizon. Current opinion in pharmacology, Vol. 12, H. 5. pp. 562-566.

Wenzler, T. and Steinhuber, A. and Wittlin, S. and Scheurer, C. and Brun, R. and Trampuz, A.. (2012) Isothermal microcalorimetry, a new tool to monitor drug action against Trypanosoma brucei and Plasmodium falciparum. PLoS neglected tropical diseases, Vol. 6, H. 6 , e1668.

Banerjee, M. and Farahat, A. A. and Kumar, A. and Wenzler, T. and Brun, R. and Munde, M. M. and Wilson, W. D. and Zhu, X. and Werbovetz, K. A. and Boykin, D. W.. (2012) Synthesis, DNA binding and antileishmanial activity of low molecular weight bis-arylimidamides. European journal of medicinal chemistry, 55. pp. 449-454.

Bakunov, S. A. and Bakunova, S. M. and Wenzler, T. and Ghebru, M. and Werbovetz, K. A. and Brun, R. and Tidwell, R. R.. (2011) Correction to synthesis and antiprotozoal activity of cationic1,4-diphenyl-1H-1,2,3-triazoles. Journal of medicinal chemistry, 54 (12). p. 4281.

Ismail, M. A. and Bialy, S. A. and Brun, R. and Wenzler, T. and Nanjunda, R. and Wilson, W. D. and Boykin, D. W.. (2011) Dicationic phenyl-2,2'-bichalcophenes and analogues as antiprotozoal agents. Bioorganic & medicinal chemistry : a Tetrahedron publication for the rapid dissemenination of full original research papers and critical reviews on biomolecular chemistry, medicinal chemistry and related disciplines, 19 (2). pp. 978-984.

Farahat, A. A. and Paliakov, E. and Kumar, A. and Barghash, A. E. and Goda, F. E. and Eisa, H. M. and Wenzler, T. and Brun, R. and Liu, Y. and Wilson, W. D. and Boykin, D. W.. (2011) Exploration of larger central ring linkers in furamidine analogues : synthesis and evaluation of their DNA binding, antiparasitic and fluorescence properties. Bioorganic & medicinal chemistry : a Tetrahedron publication for the rapid dissemenination of full original research papers and critical reviews on biomolecular chemistry, medicinal chemistry and related disciplines, 19 (7). pp. 2156-2167.

Arafa, R. K. and Wenzler, T. and Brun, R. and Chai, Y. and Wilson, D.. (2011) Molecular modeling study and synthesis of novel dicationic flexible triaryl guanidines and imidamides as antiprotozoal agents. European journal of medicinal chemistry, 46 (12). pp. 5852-5860.

Reid, C. S. and Patrick, D. A. and He, S. and Fotie, J. and Premalatha, K. and Tidwell, R. R. and Wang, M. Z. and Liu, Q. and Gershkovich, P. and Wasan, K. M. and Wenzler, T. and Brun, R. and Werbovetz, K. A.. (2011) Synthesis and antitrypanosomal evaluation of derivatives of N-benzyl-1,2-dihydroquinolin-6-ols : effect of core substitutions and salt formation. Bioorganic & medicinal chemistry : a Tetrahedron publication for the rapid dissemenination of full original research papers and critical reviews on biomolecular chemistry, medicinal chemistry and related disciplines, 19 (1). pp. 513-523.

Mosimann, M. and Goshima, S. and Wenzler, T. and Luscher, A. and Uozumi, N. and Mäser, P.. (2010) A Trk/HKT-type K+ transporter from Trypanosoma brucei. Eukaryotic Cell, Vol. 9, H. 4. pp. 539-546.

Fotie, J. and Kaiser, M. and Delfin, D. A. and Manley, J. and Reid, C. S. and Paris, J. M. and Wenzler, T. and Maes, L. and Mahasenan, K. V. and Li, C. and Werbovetz, K. A.. (2010) Antitrypanosomal activity of 1,2-dihydroquinolin-6-ols and their ester derivatives. Journal of medicinal chemistry, 53 (3). pp. 966-982.

Athri, P. and Wenzler, T. and Tidwell, R. and Bakunova, S. M. and Wilson, W. D.. (2010) Pharmacophore model for pentamidine analogs active against Plasmodium falciparum. European Journal of Medicinal Chemistry, 45 (12). pp. 6147-6151.

Branowska, D. and Farahat, A. A. and Kumar, A. and Wenzler, T. and Brun, R. and Liu, Y. and Wilson, W. D. and Boykin, D. W.. (2010) Synthesis and antiprotozoal activity of 2,5-bis[amidinoaryl]thiazoles. Bioorganic & Medicinal Chemistry, 18 (10). pp. 3551-3558.

Bakunov, S. A. and Bakunova, S. M. and Wenzler, T. and Ghebru, M. and Werbovetz, K. A. and Brun, R. and Tidwell, R. R.. (2010) Synthesis and antiprotozoal activity of cationic 1,4-diphenyl-1H-1,2,3-triazoles. Journal of Medicinal Chemistry, 53 (1). pp. 254-272.

Farahat, A. A. and Kumar, A. and Say, M. and Barghash Aedm, and Goda, F. E. and Eisa, H. M. and Wenzler, T. and Brun, R. and Liu, Y. and Mickelson, L. and Wilson, W. D. and Boykin, D. W.. (2010) Synthesis, DNA binding, fluorescence measurements and antiparasitic activity of DAPI related diamidines. Bioorganic & Medicinal Chemistry, 18 (2). pp. 557-566.

Malebo, H. M. and Wenzler, T. and Cal, M. and Swaleh, S. A. and Omolo, M. O. and Hassanali, A. and Sequin, U. and Hamburger, M. and Brun, R. and Ndiege, I. O.. (2009) Antiplasmodial, anti-trypanosomal, anti-leishmanial and cytotoxicity activity of selected Tanzanian medicinal plants. Tanzania journal of health research, Vol. 11, H. 4. pp. 226-234.

Wenzler, T. and Boykin, D. W. and Ismail, M. A. and Hall, J. E. and Tidwell, R. R. and Brun, R.. (2009) New treatment option for second stage African sleeping sickness: In vitro and in vivo efficacy of aza analogs of DB289. Antimicrobial agents and chemotherapy : AAC, Vol. 53, H. 10. pp. 4185-4192.

Bakunova, S. M. and Bakunov, S. A. and Patrick, D. A. and Kumar, E. V. and Ohemeng, K. A. and Bridges, A. S. and Wenzler, T. and Barszcz, T. and Jones, S. K. and Werbovetz, K. A. and Brun, R. and Tidwell, R. R.. (2009) Structure-activity study of pentamidine analogues as antiprotozoal agents. Journal of Medicinal Chemistry, 52 (7). pp. 2016-2035.

Hu, L. and Arafa, R. K. and Ismail, M. A. and Patel, A. and Munde, M. and Wilson, W. D. and Wenzler, T. and Brun, R. and Boykin, D. W.. (2009) Synthesis and activity of azaterphenyl diamidines against Trypanosoma brucei rhodesiense and Plasmodium falciparum. Bioorganic & medicinal chemistry letters : a Tetrahedron publication for the rapid dissemination of preliminary communications on all aspects of bioorganic chemistry, medicinal chemistry, bioinorganic chemistry and related disciplines, Vol. 17, H. 18. pp. 6651-6658.

Patrick, D. A. and Bakunov, S. A. and Bakunova, S. M. and Suresh Kumar E. V., and Chen, H. and Jones, S. K. and Wenzler, T. and Barzcz, T. and Werbovetz, K. A. and Brun, R. and Tidwell, R. R.. (2009) Synthesis and antiprotozoal activities of dicationic bis(phenoxymethyl)benzenes, bis(phenoxymethyl)naphthalenes, and bis(benzyloxy)naphthalenes. European Journal of Medicinal Chemistry, 44 (9). pp. 3543-3551.

Bakunova, S. M. and Bakunov, S. A. and Wenzler, T. and Barszcz, T. and Werbovetz, K. A. and Brun, R. and Tidwell, R. R.. (2009) Synthesis and antiprotozoal activity of pyridyl analogues of pentamidine. Journal of Medicinal Chemistry, 52 (15). pp. 4657-4667.

Bakunov, S. A. and Bakunova, S. M. and Bridges, A. S. and Wenzler, T. and Barszcz, T. and Werbovetz, K. A. and Brun, R. and Tidwell, R. R.. (2009) Synthesis and antiprotozoal properties of pentamidine congeners bearing the benzofuran motif. Journal of Medicinal Chemistry, 52 (18). pp. 5763-5767.

This list was generated on Thu Mar 28 18:52:17 2024 CET.