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Items where Author is "Mäser, P."

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Number of items: 59.

2023

Sevik Kilicaslan, O. and Cretton, S. and Hausmann, E. and Quirós-Guerrero, L. and Karimou, S. and Kaiser, M. and Mäser, P. and Christen, P. and Cuendet, M.. (2023) Antiprotozoal activity of natural products from Nigerien plants used in folk medicine. Front Pharmacol, 14. p. 1190241.

Seebacher, W. and Kaiser, M. and Mäser, P. and Saf, R. and Pferschy-Wenzig, E. M. and Weis, R.. (2023) Benzyl- and dibenzyl tetrahydropyridinylidene ammonium salts with antiplasmodial and antitrypanosomal activity. Monatshefte fuÌ�r Chemie, 154. pp. 105-114.

Rao, S. P. S. and Gould, M. K. and Noeske, J. and Saldivia, M. and Jumani, R. S. and Ng, P. S. and Rene, O. and Chen, Y. L. and Kaiser, M. and Ritchie, R. and Francisco, A. F. and Johnson, N. and Patra, D. and Cheung, H. and Deniston, C. and Schenk, A. D. and Cortopassi, W. A. and Schmidt, R. S. and Wiedemar, N. and Thomas, B. and Palkar, R. and Ghafar, N. A. and Manoharan, V. and Luu, C. and Gable, J. E. and Wan, K. F. and Myburgh, E. and Mottram, J. C. and Barnes, W. and Walker, J. and Wartchow, C. and Aziz, N. and Osborne, C. and Wagner, J. and Sarko, C. and Kelly, J. M. and Manjunatha, U. H. and Mäser, P. and Jiricek, J. and Lakshminarayana, S. B. and Barrett, M. P. and Diagana, T. T.. (2023) Cyanotriazoles are selective topoisomerase II poisons that rapidly cure trypanosome infections. Science, 380 (6652). pp. 1349-1356.

Walz, A. and Duffey, M. and Aljayyoussi, G. and Sax, S. and Leroy, D. and Besson, A. and Burrows, J. N. and Cherkaoui-Rbati, M. H. and Gobeau, N. and Westwood, M.-A. and Siethoff, C. and Gamo, S. and Mäser, P. and Wittlin, S.. (2023) The Parasite Reduction Ratio (PRR) assay version 2: standardized assessment of Plasmodium falciparum viability after antimalarial treatment in vitro. Pharmaceuticals (Basel), 16 (2). p. 163.

2022

Mousavi, A. and Foroumadi, P. and Emamgholipour, Z. and Mäser, P. and Kaiser, M. and Foroumadi, A.. (2022) 2-(Nitroaryl)-5-substituted-1,3,4-thiadiazole derivatives with antiprotozoal activities: in vitro and in vivo study. Molecules, 27. p. 5559.

Dolensky, J. and Hinteregger, C. and Leitner, A. and Seebacher, W. and Saf, R. and Belaj, F. and Mäser, P. and Kaiser, M. and Weis, R.. (2022) Antiprotozoal activity of azabicyclo-nonanes linked to tetrazole or sulfonamide cores. Molecules, 27 (19). p. 6217.

Koester, D. C. and Marx, V. M. and Williams, S. and Jiricek, J. and Dauphinais, M. and René, O. and Miller, S. L. and Zhang, L. and Patra, D. and Chen, Y. L. and Cheung, H. and Gable, J. and Lakshminarayana, S. B. and Osborne, C. and Galarneau, J. R. and Kulkarni, U. and Richmond, W. and Bretz, A. and Xiao, L. and Supek, F. and Wiesmann, C. and Honnappa, S. and Be, C. and Mäser, P. and Kaiser, M. and Ritchie, R. and Barrett, M. P. and Diagana, T. T. and Sarko, C. and Rao, S. P. S.. (2022) Discovery of novel quinoline-based proteasome inhibitors for Human African Trypanosomiasis (HAT). Journal of medicinal chemistry, 65. 11776−11787.

Scheiber, N. and Blaser, G. and Pferschy-Wenzig, E. M. and Kaiser, M. and Mäser, P. and Presser, A.. (2022) Efficient oxidative dearomatisations of substituted phenols using hypervalent iodine (iii) reagents and antiprotozoal evaluation of the resulting cyclohexadienones against T. b. rhodesiense and P. falciparum Strain NF54. Molecules, 27 (19). p. 6559.

Bernhard, S. and Kaiser, M. and Burri, C. and Mäser, P.. (2022) Fexinidazole for human African trypanosomiasis, the fruit of a successful public-private partnership. Diseases, 10 (4). p. 90.

Mäser, P.. (2022) Filariae as organisms. In: Human and animal filariases: Landscape, challenges, and control. Hoboken, New Jersey, pp. 17-32.

Sevik Kilicaslan, O. and Cretton, S. and Quiros-Guerrero, L. and Bella, M. A. and Kaiser, M. and Mäser, P. and Ndongo, J. T. and Cuendet, M.. (2022) Isolation and structural elucidation of compounds from Pleiocarpa bicarpellata and their in vitro antiprotozoal activity. Molecules, 27 (7). p. 2200.

Beilstein, S. and El Phil, R. and Sahraoui, S. S. and Scapozza, L. and Kaiser, M. and Mäser, P.. (2022) Laboratory selection of trypanosomatid pathogens for drug resistance. Pharmaceuticals (Basel), 15 (2). p. 135.

Wipf, N. C. and Duchemin, W. and Kouadio, F. A. and Fodjo, B. K. and Sadia, C. G. and Mouhamadou, C. S. and Vavassori, L. and Mäser, P. and Mavridis, K. and Vontas, J. and Müller, P.. (2022) Multi-insecticide resistant malaria vectors in the field remain susceptible to malathion, despite the presence of Ace1 point mutations. PLoS Genet, 18 (2). e1009963.

Hermann, T. and Wallner, R. and Dolensky, J. and Seebacher, W. and Pferschy-Wenzig, E. -M. and Kaiser, M. and Mäser, P. and Weis, R.. (2022) New derivatives of the multi-stage active Malaria Box compound MMV030666 and their antiplasmodial potencies. Pharmaceuticals (Basel), 15 (12). p. 1503.

Hinteregger, C. and Dolensky, J. and Seebacher, W. and Saf, R. and Mäser, P. and Kaiser, M. and Weis, R.. (2022) Synthesis and antiprotozoal activity of azabicyclo-nonane pyrimidine hybrids. Molecules, 28. p. 307.

2021

Hochegger, P. and Dolensky, J. and Seebacher, W. and Saf, R. and Kaiser, M. and Mäser, P. and Weis, R.. (2021) 8-amino-6-methoxyquinoline-tetrazole hybrids: Impact of linkers on antiplasmodial activity. Molecules, 26 (18). p. 5530.

Szabó, L. U. and Kaiser, M. and Mäser, P. and Schmidt, T. J.. (2021) Antiprotozoal Nor-triterpene alkaloids from Buxus sempervirens L. Antibiotics (Basel), 10 (6). p. 696.

Brand, M. and Wang, L. and Agnello, S. and Gazzola, S. and Gall, F. M. and Raguz, L. and Kaiser, M. and Schmidt, R. S. and Ritschl, A. and Jelk, J. and Hemphill, A. and Mäser, P. and Butikofer, P. and Adams, M. and Riedl, R.. (2021) Antiprotozoal structure-activity relationships of synthetic leucinostatin derivatives and elucidation of their mode of action. Angewandte Chemie, 60 (28). pp. 15613-15621.

Greve, H. L. and Kaiser, M. and Mäser, P. and Schmidt, T. J.. (2021) Boswellic acids show in vitro activity against Leishmania donovani. Molecules, 26 (12). p. 3651.

Rocha-Hasler, M. and de Oliveira, G. M. and da Gama, A. N. and Fiuza, L. F. A. and Fesser, A. F. and Cal, M. and Rocchetti, R. and Peres, R. B. and Guan, X. L. and Kaiser, M. and Soeiro, M. N. C. and Mäser, P.. (2021) Combination with tomatidine improves the potency of posaconazole against Trypanosoma cruzi. Front Cell Infect Microbiol, 11. p. 617917.

Boberg, M. and Cal, M. and Kaiser, M. and Jansson-Lofmark, R. and Mäser, P. and Ashton, M.. (2021) Enantiospecific antitrypanosomal in vitro activity of eflornithine. PLoS Negl Trop Dis, 15 (7). e0009583.

Wittlin, S. and Mäser, P.. (2021) From magic bullet to magic bomb: reductive bioactivation of antiparasitic agents. ACS Infect Dis, 7 (10). pp. 2777-2786.

Cretton, S. and Genta-Jouve, G. and Kaiser, M. and Mäser, P. and Muñoz, O. and Bürgi, T. and Cuendet, M. and Christen, P.. (2021) Hygroline derivatives from Schizanthus tricolor and their anti-trypanosomatid and antiplasmodial activities. Phytochemistry, 192. p. 112957.

Szabó, L. U. and Kaiser, M. and Mäser, P. and Schmidt, T. J.. (2021) Identification of antiprotozoal compounds from Buxus sempervirens L. by PLS-prediction. Molecules, 26 (20). p. 6181.

Barth-Jaeggi, T. and Mäser, P.. (2021) Leishmaniasis in Europe and Central Asia: epidemiology, impact of habitat and lifestyle changes, HIV coinfection. In: Neglected tropical diseases - Europe and Central Asia. Cham, pp. 83-100.

Seebacher, W. and Mohsin, N. U. A. and Dolensky, J. and Hochegger, P. and Kaiser, M. and Mäser, P. and Saf, R. and Schuster, D. and Temml, V. and Weis, R.. (2021) Modifications and hybrids of 1,2,3,4‑tetrahydropyridinium salts and their antiprotozoal potencies. Monatshefte fuÌ�r Chemie, 152. pp. 1347-1359.

Fesser, A. and Kaiser, M. and Mäser, P.. (2021) Neue Parameter für die Wirkstofftestung gegen Trypanosoma cruzi. Biospektrum (Heidelb), 27 (2). pp. 168-170.

Hermann, T. and Hochegger, P. and Dolensky, J. and Seebacher, W. and Saf, R. and Kaiser, M. and Mäser, P. and Weis, R.. (2021) New acyl derivatives of 3-aminofurazanes and their antiplasmodial activities. Pharmaceuticals (Basel), 14 (5). p. 412.

Mahmoud, A. B. and Abd Algaffar, S. and van de Sande, W. and Khalid, S. and Kaiser, M. and Mäser, P.. (2021) Niclosamide is active in vitro against mycetoma pathogens. Molecules, 26 (13). p. 4005.

Llurba Montesino, N. and Kaiser, M. and Mäser, P. and Schmidt, T. J.. (2021) Nucleic acid amplification techniques for the detection of Schistosoma mansoni infection in humans and the intermediate snail host: a structured review and meta-analysis of diagnostic accuracy. Molecules, 26 (11). p. 3226.

Petritsch, M. and Seebacher, W. and Mohsin, N. U. and Dolensky, J. and Hochegger, P. and Kaiser, M. and Mäser, P. and Belaj, F. and Saf, R. and Kretschmer, N. and Alajlani, M. and Brantner, A. and Bauer, R. and Schuhly, W. and Weis, R.. (2021) Preparation of new 1,3-dibenzyl tetrahydropyridinylidene ammonium salts and their antimicrobial and anticellular activities. Eur J Med Chem, 210. p. 112969.

Zeelen, J. and van Straaten, M. and Verdi, J. and Hempelmann, A. and Hashemi, H. and Perez, K. and Jeffrey, P. D. and Hälg, S. and Wiedemar, N. and Mäser, P. and Papavasiliou, F. N. and Stebbins, C. E.. (2021) Structure of trypanosome coat protein VSGsur and function in suramin resistance. Nat Microbiol, 6 (3). pp. 392-400.

Hermann, T. and Hochegger, P. and Dolensky, J. and Seebacher, W. and Pferschy-Wenzig, E. M. and Saf, R. and Kaiser, M. and Mäser, P. and Weis, R.. (2021) Synthesis and structure-activity relationships of new 2-phenoxybenzamides with antiplasmodial activity. Pharmaceuticals (Basel), 14. p. 1109.

Hitz, E. and Wiedemar, N. and Passecker, A. and Graça, B. A. S. and Scheurer, C. and Wittlin, S. and Brancucci, N. M. B. and Vakonakis, I. and Mäser, P. and Voss, T. S.. (2021) The 3-phosphoinositide-dependent protein kinase 1 is an essential upstream activator of protein kinase A in malaria parasites. PLoS Biol, 19 (12). e3001483.

Flittner, D. and Kaiser, M. and Mäser, P. and Lopes, N. P. and Schmidt, T. J.. (2021) The alkaloid-enriched fraction of; The alkaloid-enriched fraction of Pachysandra terminalis (Buxaceae) shows prominent activity against Trypanosoma brucei rhodesiensePachysandra terminalis; (Buxaceae) shows prominent activity against; Trypanosoma brucei rhodesiense. Molecules, 26 (3). p. 591.

Hoffelner, M. H. and Seebacher, W. and Kaiser, M. and Mäser, P. and Pferschy-Wenzig, E. M. and Saf, R. and Belaj, F. and Kretschmer, N. and Alajlani, M. and Brantner, A. and Bauer, R. and Weis, R.. (2021) Unexpected ring‑opening of 2,3‑dihydropyridines. Monatshefte für Chemie, 152. pp. 1347-1359.

2020

Kaiser, M. and Mäser, P.. (2020) In Vitro drug efficacy testing against Trypanosoma brucei. New York.

Hoffelner, M. and Hassan, U. and Seebacher, W. and Dolensky, J. and Hochegger, P. and Kaiser, M. and Mäser, P. and Saf, R. and Weis, R.. (2020) New 2‑aminopyrimidine derivatives and their antitrypanosomal and antiplasmodial activities. Monatshefte für Chemie, 151. pp. 1375-1385.

Cretton, S. and Kaiser, M. and Karimou, S. and Ebrahimi, S. N. and Mäser, P. and Cuendet, M. and Christen, P.. (2020) Pyridine-4(1H)-one alkaloids from Waltheria indica as antitrypanosomatid agents. Journal of natural products, 83 (11). pp. 3363-3371.

2019

Walz, A. and Leroy, D. and Andenmatten, N. and Mäser, P. and Wittlin, S.. (2019) Anti-malarial ozonides OZ439 and OZ609 tested at clinically relevant compound exposure parameters in a novel ring-stage survival assay. Malaria journal, 18. p. 427.

Mäser, P.. (2019) Parasiten machen Geschichte. In: Gespräche im Garten: Kultur - Natur - Gutes Leben: Tusculum auf Mapprach. Basel, pp. 127-131.

Mohsin, N. U. A. and Seebacher, W. and Hochegger, P. and Faist, J. and Saf, R. and Kaiser, M. and Mäser, P. and Weis, R.. (2019) Synthesis of new 1-benzyl tetrahydropyridin-4-ylidene piperidinium salts and their antiplasmodial and antitrypanosomal activities. Medicinal chemistry research, 28 (5). pp. 742-753.

2018

Gysin, M. and Braissant, O. and Gillingwater, K. and Brun, R. and Mäser, P. and Wenzler, T.. (2018) Isothermal microcalorimetry - a quantitative method to monitor Trypanosoma congolense growth and growth inhibition by trypanocidal drugs in real time. International journal for parasitology. Drugs and drug resistance, 8 (2). pp. 159-164.

Mohsin, N. U. A. and Seebacher, W. and Faist, J. and Kretschmer, N. and Bauer, R. and Saf, R. and Kaiser, M. and Mäser, P. and Weis, R.. (2018) Modifications on tetrahydropyridin-4-ylidene ammonium salts and their antiprotozoal activities. Monatshefte für Chemie, 149 (4). pp. 801-812.

Mohsin, N. U. A. and Seebacher, W. and Faist, J. and Hochegger, P. and Kaiser, M. and Mäser, P. and Saf, R. and Weis, R.. (2018) The antiplasmodial and antitrypanosomal activities of novel piperazine derivatives of 3-azabicyclo[3.2.2]nonanes. Monatshefte für Chemie, 149 (1). pp. 99-109.

2017

Dawidowski, M. and Emmanouilidis, L. and Kalel, V. C. and Tripsianes, K. and Schorpp, K. and Hadian, K. and Kaiser, M. and Mäser, P. and Kolonko, M. and Tanghe, S. and Rodriguez, A. and Schliebs, W. and Erdmann, R. and Sattler, M. and Popowicz, G. M.. (2017) Inhibitors of PEX14 disrupt protein import into glycosomes and kill Trypanosoma parasites. Science, 355 (6332). pp. 1416-1420.

Seebacher, W. and Belaj, F. and Faist, J. and Saf, R. and Bucar, F. and Turek, I. and Branter, A. and Alajlani, M. and Kaiser, M. and Mäser, P. and Weis, R.. (2017) Synthesis of new pyrido-benzodiazepine salts and their antimicrobial activities. Monatshefte für Chemie, 148 (2). pp. 263-274.

2013

Ali, J. A. M. and Creek, D. J. and Burgess, K. and Allison, H. C. and Field, M. C. and Mäser, P. and de Koning, H. P.. (2013) Pyrimidine salvage in Trypanosoma brucei bloodstream forms and the trypanocidal action of halogenated pyrimidines. Molecular pharmacology : an international journal, Vol. 83, H. 2. pp. 439-453.

2012

Mäser, P. and Wittlin, S. and Rottmann, M. and Wenzler, T. and Kaiser, M. and Brun, R.. (2012) Antiparasitic agents : new drugs on the horizon. Current opinion in pharmacology, Vol. 12, H. 5. pp. 562-566.

Godel, C. and Kumar, S. and Koutsovoulos, G. and Ludin, P. and Nilsson, D. and Comandatore, F. and Wrobel, N. and Thompson, M. and Schmid, C. D. and Goto, S. and Bringaud, F. and Wolstenholme, A. and Bandi, C. and Epe, C. and Kaminsky, R. and Blaxter, M. and Mäser, P.. (2012) The genome of the heartworm, Dirofilaria immitis, reveals drug and vaccine targets. The FASEB Journal : official publication of the Federation of American Societies for Experimental Biology, Vol. 26, H. 11. pp. 4650-4661.

Gonzalez-Salgado, A. and Steinmann, M. E. and Greganova, E. and Rauch, M. and Mäser, P. and Sigel, E. and Bütikofer, P.. (2012) myo-inositol uptake is essential for bulk inositol phospholipid but not glycosylphosphatidylinositol synthesis in Trypanosoma brucei. Journal of biological chemistry, Vol. 287, H. 16. pp. 13313-13323.

2011

Ludin, P. and Nilsson, D. and Mäser, P.. (2011) Genome-wide identification of molecular mimicry candidates in parasites. PLoS ONE, 6 (3). e17546.

Lamprea-Burgunder, E. and Ludin, P. and Mäser, P.. (2011) Species-specific typing of DNA based on palindrome frequency patterns. DNA research, 18 (2). pp. 117-124.

Teka, I. A. and Kazibwe, A. J. N. and El-Sabbagh N., and Al-Salabi M. I., and Ward, C. P. and Eze, A. A. and Munday, J. C. and Mäser, P. and Matovu, E. and Barrett, M. P. and de Koning H. P., . (2011) The diamidine diminazene aceturate is a substrate for the high-affinity pentamidine transporter: implications for the development of high resistance levels in trypanosomes. Molecular pharmacology : an international journal, Vol. 80, H. 1. pp. 110-116.

2010

Mosimann, M. and Goshima, S. and Wenzler, T. and Luscher, A. and Uozumi, N. and Mäser, P.. (2010) A Trk/HKT-type K+ transporter from Trypanosoma brucei. Eukaryotic Cell, Vol. 9, H. 4. pp. 539-546.

Nerima, B. and Nilsson, D. and Mäser, P.. (2010) Comparative genomics of metabolic networks of free-living and parasitic eukaryotes. BMC Genomics, Vol. 11 , 217.

Rufener, L. and Baur, R. and Kaminsky, R. and Mäser, P. and Sigel, E.. (2010) Monepantel allosterically activates DEG-3/DES-2 channels of the gastrointestinal nematode Haemonchus contortus. Molecular pharmacology : an international journal, Vol. 78, H. 5. pp. 895-902.

Rufener, L. and Keiser, J. and Kaminsky, R. and Mäser, P. and Nilsson, D.. (2010) Phylogenomics of ligand-gated ion channels predicts monepantel effect. PLoS Pathogens, Vol. 6, H. 9 , e1001091.

2009

Kuettel, S. and Mosimann, M. and Mäser, P. and Kaiser, M. and Brun, R. and Scapozza, L. and Perozzo, R.. (2009) Adenosine kinase of T. b. Rhodesiense identified as the putative target of 4-[5-(4-phenoxyphenyl)-2H-pyrazol-3-yl]morpholine using chemical proteomics. PLoS Neglected Tropical Diseases, Vol. 3, H. 8 , e506.

This list was generated on Fri Mar 29 10:16:55 2024 CET.