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Items where Author is "Kaiser, Marcel"

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Number of items: 194.

2021

Bevkal, Shubha and Naguleswaran, Arunasalam and Rehmann, Ruth and Kaiser, Marcel and Heller, Manfred and Roditi, Isabel. (2021) An Alba-domain protein required for proteome remodelling during trypanosome differentiation and host transition. PLoS Pathogens, 17. e1009239.

2020

Bernal, Freddy A. and Gerhards, Marcel and Kaiser, Marcel and Wünsch, Bernhard and Schmidt, Thomas J.. (2020) (+/-)-trans-2-phenyl-2,3-dihydrobenzofurans as leishmanicidal agents: synthesis, in vitro evaluation and SAR analysis. European journal of medicinal chemistry, 205. p. 112493.

Hagen, James P. and Darner, Grant and Anderson, Samuel and Higgins, Katie and Leas, Derek A. and Mitra, Ananya and Mashinson, Victoria and Wol, Tasloach and Vera-Esquivel, Carlos and Belter, Bret and Cal, Monica and Kaiser, Marcel and Wallick, Alexander and Warner, Rosalie C. and Davis, Paul H.. (2020) Activity of diphenyl ether benzyl amines against Human African Trypanosomiasis. Bioorganic chemistry, 97. p. 103590.

Rao, Srinivasa P. S. and Lakshminarayana, Suresh B. and Jiricek, Jan and Kaiser, Marcel and Ritchie, Ryan and Myburgh, Elmarie and Supek, Frantisek and Tuntland, Tove and Nagle, Advait and Molteni, Valentina and Mäser, Pascal and Mottram, Jeremy C. and Barrett, Michael P. and Diagana, Thierry T.. (2020) Anti-trypanosomal proteasome inhibitors cure hemolymphatic and meningoencephalic murine infection models of african trypanosomiasis. Tropical medicine and infectious disease, 5. p. 28.

Zadali, Reza and Ebrahimi, Samad Nejad and Tofighi, Zahra and Es-haghi, Ali and Hamburger, Matthias and Kaiser, Marcel and D'Ambola, Massimiliano and De Tommasi, Nunziatina and Hadjiakhoondi, Abbas. (2020) Antiprotozoal activity of diterpenoids isolated from Zhumeria majdae - absolute configuration by circular dichroism. DARU Journal of Pharmaceutical Sciences, 28 (2). pp. 455-462.

Tasdemir, Deniz and MacIntosh, Andrew J. J. and Stergiou, Polyxeni and Kaiser, Marcel and Mansour, Nuha R. and Bickle, Quentin and Huffman, Michael A.. (2020) Antiprotozoal and antihelminthic properties of plants ingested by wild Japanese macaques (Macaca fuscata yakui) in Yakushima Island. Journal of Ethnopharmacology, 247. p. 112270.

Harrison, Justin R. and Sarkar, Sandipan and Hampton, Shahienaz and Riley, Jennifer and Stojanovski, Laste and Sahlberg, Christer and Appelqvist, Pia and Erath, Jessey and Mathan, Vinodhini and Rodriguez, Ana and Kaiser, Marcel and Pacanowska, Dolores Gonzalez and Read, Kevin D. and Johansson, Nils Gunnar and Gilbert, Ian H.. (2020) Discovery and optimization of a compound series active against Trypanosoma cruzi, the causative agent of chagas disease. Journal of medicinal chemistry, 63 (6). pp. 3066-3089.

Ponzi, Simona and Bresciani, Alberto and Kaiser, Marcel and Nardi, Valentina and Nizi, Emanuela and Ontoria, Jesus M. and Pace, Paola and Paonessa, Giacomo and Summa, Vincenzo and Harper, Steven. (2020) Discovery of 4-((1-(1H-imidazol-2-yl)alkoxy)methyl)pyridines as a new class of Trypanosoma cruzi growth inhibitors. Bioorganic & medicinal chemistry letters, 30 (8). p. 127052.

Mahmoud, Abdelhalim Babiker and Danton, Ombeline and Kaiser, Marcel and Khalid, Sami and Hamburger, Matthias and Mäser, Pascal. (2020) HPLC-based activity profiling for antiprotozoal compounds in Croton gratissimus and Cuscuta hyalina. Frontiers in Pharmacology, 11. p. 1246.

Greve, Hippolyt L. and Kaiser, Marcel and Schmidt, Thomas J.. (2020) Investigation of antiplasmodial effects of terpenoid compounds isolated from myrrh. Planta medica, 86 (9). pp. 643-654.

Mahmoud, Abdelhalim Babiker and Danton, Ombeline and Kaiser, Marcel and Han, Sohee and Moreno, Aitor and Abd Algaffar, Shereen and Khalid, Sami and Oh, Won Keun and Hamburger, Matthias and Mäser, Pascal. (2020) Lignans, amides, and saponins from Haplophyllum tuberculatum and their antiprotozoal activity. Molecules, 25 (12). p. 2825.

Mahmoud, Abdelhalim Babiker and Mäser, Pascal and Kaiser, Marcel and Hamburger, Matthias and Khalid, Sami. (2020) Mining sudanese medicinal plants for antiprotozoal agents. Frontiers in pharmacology, 11. p. 865.

Fesser, Anna F. and Braissant, Olivier and Olmo, Francisco and Kelly, John M. and Mäser, Pascal and Kaiser, Marcel. (2020) Non-invasive monitoring of drug action: a new live in vitro assay design for Chagas' disease drug discovery. PLoS Neglected Tropical Diseases, 14 (7). e0008487.

Dawidowski, Maciej and Kalel, Vishal C. and Napolitano, Valeria and Fino, Roberto and Schorpp, Kenji and Emmanouilidis, Leonidas and Lenhart, Dominik and Ostertag, Michael and Kaiser, Marcel and Kolonko, Marta and Tippler, Bettina and Schliebs, Wolfgang and Dubin, Grzegorz and Mäser, Pascal and Tetko, Igor V. and Hadian, Kamyar and Plettenburg, Oliver and Erdmann, Ralf and Sattler, Michael and Popowicz, Grzegorz M.. (2020) Structure-activity relationship in pyrazolo[4,3-c]pyridines, first inhibitors of PEX14-PEX5 protein-protein interaction with trypanocidal activity. Journal of medicinal chemistry, 63 (2). pp. 847-879.

Bernal, Freddy A. and Kaiser, Marcel and Wünsch, Bernhard and Schmidt, Thomas J.. (2020) Structure-activity relationships of cinnamate ester analogues as potent antiprotozoal agents. ChemMedChem, 15. pp. 68-78.

2019

Shi, Yan-Ni and Pusch, Stefan and Shi, Yi-Ming and Richter, Christian and Maciá-Vicente, Jose G. and Schwalbe, Harald and Kaiser, Marcel and Opatz, Till and Bode, Helge B.. (2019) (+/-)-Alternarlactones A and B, two antiparasitic alternariol-like dimers from the fungus Alternaria alternata p1210 isolated from the halophyte Salicornia sp. Journal of Organic Chemistry, 84 (17). pp. 11203-11209.

Fayez, Shaimaa and Li, Jun and Feineis, Doris and Aké Assi, Laurent and Kaiser, Marcel and Brun, Reto and Anany, Mohamed A. and Wajant, Harald and Bringmann, Gerhard. (2019) A Near-Complete Series of Four Atropisomeric Jozimine A; 2; -Type Naphthylisoquinoline Dimers with Antiplasmodial and Cytotoxic Activities and Related Alkaloids from; Ancistrocladus abbreviatus;. Journal of natural products, 82 (11). pp. 3033-3046.

Tshitenge, Dieudonné Tshitenge and Bruhn, Torsten and Feineis, Doris and Mudogo, Virima and Kaiser, Marcel and Brun, Reto and Bringmann, Gerhard. (2019) An unusually broad series of seven cyclombandakamines, bridged dimeric naphthylisoquinoline alkaloids from the congolese liana ancistrocladus ealaensis. Scientific reports, 9. p. 9812.

Hochegger, Patrick and Faist, Johanna and Seebacher, Werner and Saf, Robert and Mäser, Pascal and Kaiser, Marcel and Weis, Robert. (2019) Antiprotozoal activities of tetrazole-quinolines with aminopiperidine linker. Medicinal chemistry (Shariqah (United Arab Emirates)), 15 (4). pp. 409-416.

Mofidi Tabatabaei, Sahar and Nejad Ebrahimi, Samad and Salehi, Peyman and Sonboli, Ali and Tabefam, Marzieh and Kaiser, Marcel and Hamburger, Matthias and Moridi Farimani, Mahdi. (2019) Antiprotozoal germacranolide sesquiterpene lactones from Tanacetum sonbolii. Planta medica, 85 (5). pp. 424-430.

Galkina, Anna and Krause, Nico and Lenz, Mairin and Daniliuc, Constantin G. and Kaiser, Marcel and Schmidt, Thomas J.. (2019) Antitrypanosomal activity of sesquiterpene lactones from Helianthus tuberosus L. including a new furanoheliangolide with an unusual structure. Molecules, 24 (6). p. 1068.

Saccoliti, Francesco and Madia, Valentina Noemi and Tudino, Valeria and De Leo, Alessandro and Pescatori, Luca and Messore, Antonella and De Vita, Daniela and Scipione, Luigi and Brun, Reto and Kaiser, Marcel and Mäser, Pascal and Calvet Alvarez, Claudia Magalhaes and Jennings, Gareth K. and Podust, Larissa M. and Pepe, Giacomo and Cirilli, Roberto and Faggi, Cristina and Di Marco, Annalise and Battista, Maria Rosaria and Summa, Vincenzo and Costi, Roberta and Di Santo, Roberto. (2019) Design, synthesis, and biological evaluation of new 1-(Aryl-1H-pyrrolyl)(phenyl)methyl-1H-imidazole derivatives as antiprotozoal agents. Journal of Medicinal Chemistry, 62 (3). pp. 1330-1347.

Tshitenge, Dieudonné Tshitenge and Bruhn, Torsten and Feineis, Doris and Schmidt, David and Mudogo, Virima and Kaiser, Marcel and Brun, Reto and Würthner, Frank and Awale, Suresh and Bringmann, Gerhard. (2019) Ealamines A-H, a Series of Naphthylisoquinolines with the Rare 7,8'-Coupling Site, from the Congolese Liana; Ancistrocladus ealaensis; , Targeting Pancreatic Cancer Cells. Journal of natural products, 82 (11). pp. 3150-3164.

Babanezhad Harikandei, Kosar and Salehi, Peyman and Ebrahimi, Samad Nejad and Bararjanian, Morteza and Kaiser, Marcel and Khavasi, Hamid Reza and Al-Harrasi, Ahmed. (2019) N-substituted noscapine derivatives as new antiprotozoal agents: synthesis, antiparasitic activity and molecular docking study. Bioorganic chemistry, 91. p. 103116.

Kimani, Njogu M. and Backhaus, Solveig and Matasyoh, Josphat C. and Kaiser, Marcel and Herrmann, Fabian C. and Schmidt, Thomas J. and Langer, Klaus. (2019) Preparation of sesquiterpene lactone-loaded pla nanoparticles and evaluation of their antitrypanosomal activity. Molecules, 24 (11). E2110.

Hochegger, Patrick and Faist, Johanna and Seebacher, Werner and Saf, Robert and Mäser, Pascal and Kaiser, Marcel and Weis, Robert. (2019) Synthesis and structure-activity relationships for new 6-fluoroquinoline derivatives with antiplasmodial activity. Bioorganic & medicinal chemistry, 27 (10). pp. 2052-2065.

De Gasparo, Raoul and Halgas, Ondrej and Harangozo, Dora and Kaiser, Marcel and Pai, Emil F. and Krauth-Siegel, R. Luise and Diederich, François. (2019) Targeting a large active site : structure-based design of nanomolar inhibitors of Trypanosoma brucei trypanothione reductase. Chemistry - A European Journal, 25 (49). pp. 11416-11421.

2018

Giroud, Maude and Kuhn, Bernd and Saint-Auret, Sarah and Kuratli, Christoph and Martin, Rainer E. and Schuler, Franz and Diederich, François and Kaiser, Marcel and Brun, Reto and Schirmeister, Tanja and Haap, Wolfgang. (2018) 2 H-1,2,3-Triazole-based dipeptidyl nitriles : potent, selective, and Trypanocidal rhodesain inhibitors by structure-based design. Journal of medicinal chemistry, 61 (8). pp. 3370-3388.

Cretton, Sylvian and Oyarzún, Alejandra and Righi, Davide and Sahib, Lamia and Kaiser, Marcel and Christen, Philippe and Fajardo, Victor. (2018) A new antifungal and antiprotozoal bibenzyl derivative from Gavilea lutea. Natural Product Research, 32 (6). pp. 695-701.

Fayez, Shaimaa and Feineis, Doris and Aké Assi, Laurent and Kaiser, Marcel and Brun, Reto and Awale, Suresh and Bringmann, Gerhard. (2018) Ancistrobrevines E-J and related naphthylisoquinoline alkaloids from the West African liana Ancistrocladus abbreviatus with inhibitory activities against Plasmodium falciparum and PANC-1 human pancreatic cancer cells. Fitoterapia, 131. pp. 245-259.

Royo, Santiago and Schirmeister, Tanja and Kaiser, Marcel and Jung, Sascha and Rodríguez, Santiago and Bautista, José Manuel and González, Florenci V.. (2018) Antiprotozoal and cysteine proteases inhibitory activity of dipeptidyl enoates. Bioorganic & medicinal chemistry, 26 (16). pp. 4624-4634.

Tabefam, Marzieh and Moridi Farimani, Mahdi and Danton, Ombeline and Ramseyer, Justine and Kaiser, Marcel and Ebrahimi, Samad Nejad and Salehi, Peyman and Batooli, Hoosien and Potterat, Olivier and Hamburger, Matthias. (2018) Antiprotozoal diterpenes from Perovskia abrotanoides. Planta Medica, 84 (12-13). pp. 913-919.

Kimani, Njogu M. and Matasyoh, Josphat C. and Kaiser, Marcel and Brun, Reto and Schmidt, Thomas J.. (2018) Antiprotozoal sesquiterpene lactones and other constituents from Tarchonanthus camphoratus and Schkuhria pinnata. Journal of natural products, 81 (1). pp. 124-130.

Saccoliti, Francesco and Madia, Valentina Noemi and Tudino, Valeria and De Leo, Alessandro and Pescatori, Luca and Messore, Antonella and De Vita, Daniela and Scipione, Luigi and Brun, Reto and Kaiser, Marcel and Mäser, Pascal and Calvet, Claudia Magalhaes and Jennings, Gareth K. and Podust, Larissa M. and Costi, Roberta and Di Santo, Roberto. (2018) Biological evaluation and structure-activity relationships of imidazole-based compounds as antiprotozoal agents. European journal of medicinal chemistry, 156. pp. 53-60.

De Gasparo, Raoul and Brodbeck-Persch, Elke and Bryson, Steve and Hentzen, Nina B. and Kaiser, Marcel and Pai, Emil F. and Krauth-Siegel, R. Luise and Diederich, François. (2018) Biological evaluation and x-ray co-crystal structures of cyclohexylpyrrolidine ligands for trypanothione reductase, an enzyme from the redox metabolism of trypanosoma. ChemMedChem, 13 (9). pp. 957-967.

O' Donovan, Daniel H. and Aillard, Paul and Berger, Martin and de la Torre, Aurélien and Petkova, Desislava and Knittl-Frank, Christian and Geerdink, Danny and Kaiser, Marcel and Maulide, Nuno. (2018) C-H activation enables a concise total synthesis of quinine and analogues with enhanced antimalarial activity. Angewandte Chemie (International ed. in English), 57 (33). pp. 10737-10741.

Wesche, Frank and Adihou, Hélène and Kaiser, Astrid and Wurglics, Mario and Schubert-Zsilavecz, Manfred and Kaiser, Marcel and Bode, Helge B.. (2018) Combined approach of backbone amide linking and on-resin n-methylation for the synthesis of bioactive and metabolically stable peptides. Journal of medicinal chemistry, 61 (9). pp. 3930-3938.

Kimani, Njogu M. and Matasyoh, Josphat C. and Kaiser, Marcel and Nogueira, Mauro S. and Trossini, Gustavo H. G. and Schmidt, Thomas J.. (2018) Complementary quantitative structure-activity relationship models for the antitrypanosomal activity of sesquiterpene lactones. International journal of molecular sciences, 19 (12). p. 3271.

Uliassi, Elisa and Piazzi, Lorna and Belluti, Federica and Mazzanti, Andrea and Kaiser, Marcel and Brun, Reto and Moraes, Carolina B. and Freitas-Junior, Lucio H. and Gul, Sheraz and Kuzikov, Maria and Ellinger, Bernhard and Borsari, Chiara and Costi, Maria Paola and Bolognesi, Maria Laura. (2018) Development of a focused library of triazole-linked privileged-structure-based conjugates leading to the discovery of novel phenotypic hits against protozoan parasitic infections. ChemMedChem, 13 (7). pp. 678-683.

Ferrigno, Federica and Biancofiore, Ilaria and Malancona, Savina and Ponzi, Simona and Paonessa, Giacomo and Graziani, Rita and Bresciani, Alberto and Gennari, Nadia and Di Marco, Annalise and Kaiser, Marcel and Summa, Vincenzo and Harper, Steven and Ontoria, Jesus M.. (2018) Discovery of 2-(1H-imidazo-2-yl)piperazines as a new class of potent and non-cytotoxic inhibitors of Trypanosoma brucei growth in vitro. Bioorganic & medicinal chemistry letters, 28 (23-24). pp. 3689-3692.

Zhang, Huaisheng and Collins, Jasmine and Nyamwihura, Rogers and Ware, Shelbi and Kaiser, Marcel and Ogungbe, Ifedayo Victor. (2018) Discovery of a quinoline-based phenyl sulfone derivative as an antitrypanosomal agent. Bioorganic & medicinal chemistry, 28 (9). pp. 1647-1651.

Ebiloma, Godwin U. and Ayuga, Teresa Díaz and Balogun, Emmanuel O. and Gil, Lucía Abad and Donachie, Anne and Kaiser, Marcel and Herraiz, Tomás and Inaoka, Daniel K. and Shiba, Tomoo and Harada, Shigeharu and Kita, Kiyoshi and de Koning, Harry P. and Dardonville, Christophe. (2018) Inhibition of trypanosome alternative oxidase without its N-terminal mitochondrial targeting signal (ΔMTS-TAO) by cationic and non-cationic 4-hydroxybenzoate and 4-alkoxybenzaldehyde derivatives active against T. brucei and T. congolense. European journal of medicinal chemistry, 150. pp. 385-402.

Levatić, Jurica and Pavić, Kristina and Perković, Ivana and Uzelac, Lidija and Ester, Katja and Kralj, Marijeta and Kaiser, Marcel and Rottmann, Matthias and Supek, Fran and Zorc, Branka. (2018) Machine learning prioritizes synthesis of primaquine ureidoamides with high antimalarial activity and attenuated cytotoxicity. European journal of medicinal chemistry, 146. pp. 651-667.

Tshitenge, Dieudonné Tshitenge and Feineis, Doris and Mudogo, Virima and Kaiser, Marcel and Brun, Reto and Seo, Ean-Jeong and Efferth, Thomas and Bringmann, Gerhard. (2018) Mbandakamine-type naphthylisoquinoline dimers and related alkaloids from the central African liana ancistrocladus ealaensis with antiparasitic and antileukemic activities. Journal of natural products, 81 (4). pp. 918-933.

Zhao, Lei and Cai, Xiaofeng and Kaiser, Marcel and Bode, Helge B.. (2018) Methionine-containing rhabdopeptide/xenortide-like peptides from heterologous expression of the biosynthetic gene cluster kj12ABC in Escherichia coli. Journal of natural products, 81 (10). pp. 2292-2295.

Tallini, Luciana R. and Torras-Claveria, Laura and Borges, Warley de Souza and Kaiser, Marcel and Viladomat, Francesc and Zuanazzi, José Angelo S. and Bastida, Jaume. (2018) N-oxide alkaloids from Crinum amabile (Amaryllidaceae). Molecules, 23 (6). E1277.

Farimani, Mahdi Moridi and Khodaei, Bahareh and Moradi, Hanzaleh and Aliabadi, Abbas and Ebrahimi, Samad Nejad and De Mieri, Maria and Kaiser, Marcel and Hamburger, Matthias. (2018) Phytochemical study of Salvia leeriifolia roots: rearranged abietane diterpenoids with antiprotozoal activity. Journal of Natural Products, 81 (6). pp. 1384-1390.

Farimani, Mahdi M. and Khodaei, Bahareh and Moradi, Hanzaleh and Aliabadi, Abbas and Ebrahimi, Samad N. and De Mieri, Maria and Kaiser, Marcel and Hamburger, Matthias. (2018) Phytochemical study of Salvia leriifolia roots : rearranged abietane diterpenoids with antiprotozoal activity. Journal of natural products, 81 (6). pp. 1384-1390.

Guo, Huijuan and Schmidt, Alexander and Stephan, Philipp and Raguž, Luka and Braga, Daniel and Kaiser, Marcel and Dahse, Hans-Martin and Weigel, Christiane and Lackner, Gerald and Beemelmanns, Christine. (2018) Precursor-directed diversification of cyclic tetrapeptidic pseudoxylallemycins. ChemBioChem, 19 (21). pp. 2307-2311.

Giroud, Maude and Dietzel, Uwe and Anselm, Lilli and Banner, David and Kuglstatter, Andreas and Benz, Jörg and Blanc, Jean-Baptiste and Gaufreteau, Delphine and Liu, Haixia and Lin, Xianfeng and Stich, August and Kuhn, Bernd and Schuler, Franz and Kaiser, Marcel and Brun, Reto and Schirmeister, Tanja and Kisker, Caroline and Diederich, François and Haap, Wolfgang. (2018) Repurposing a library of human cathepsin L ligands : identification of macrocyclic lactams as potent rhodesain and Trypanosoma brucei inhibitors. Journal of medicinal chemistry, 61 (8). pp. 3350-3369.

Zhao, Lei and Kaiser, Marcel and Bode, Helge B.. (2018) Rhabdopeptide/Xenortide-like peptides from Xenorhabdus innexi with terminal amines showing potent antiprotozoal activity. Organic Letters, 20 (17). pp. 5116-5120.

Kimani, Njogu M. and Matasyoh, Josphat C. and Kaiser, Marcel and Brun, Reto and Schmidt, Thomas J.. (2018) Sesquiterpene lactones from Vernonia cinerascens sch. bip. and their in vitro antitrypanosomal activity. Molecules: A Journal of Synthetic Chemistry and Natural Product Chemistry , 23 (2). E248.

Presser, Armin and Lainer, Gunda and Kretschmer, Nadine and Schuehly, Wolfgang and Saf, Robert and Kaiser, Marcel and Kalt, Marc-Manuel. (2018) Synthesis of jacaranone-derived nitrogenous cyclohexadienones and their antiproliferative and antiprotozoal activities. Molecules, 23 (11). E2902.

Krieger, Johannes and Smeilus, Toni and Kaiser, Marcel and Seo, Ean-Jeong and Efferth, Thomas and Giannis, Athanassios. (2018) Total synthesis and biological investigation of (-)-artemisinin : the antimalarial activity of artemisinin is not stereospecific. Angewandte Chemie, 57 (27). pp. 8293-8296.

2017

Tallini, Luciana R. and Andrade, Jean Paulo de and Kaiser, Marcel and Viladomat, Francesc and Nair, Jerald J. and Zuanazzi, José Angelo S. and Bastida, Jaume. (2017) Alkaloid constituents of the amaryllidaceae plant amaryllis belladonna L. Molecules, 22 (9). p. 1437.

Althaus, Julia B. and Malyszek, Claudine and Kaiser, Marcel and Brun, Reto and Schmidt, Thomas J.. (2017) Alkamides from Anacyclus pyrethrum L. and their in vitro antiprotozoal activity. Molecules, 22 (5). p. 796.

Kimani, Njogu M. and Matasyoh, Josphat C. and Kaiser, Marcel and Brun, Reto and Schmidt, Thomas J.. (2017) Anti-trypanosomatid elemanolide sesquiterpene lactones from Vernonia lasiopus O. Hoffm. Molecules, 22 (4). E597.

Bringmann, Gerhard and Seupel, Raina and Feineis, Doris and Xu, Minjuan and Zhang, Guoliang and Kaiser, Marcel and Brun, Reto and Seo, Ean-Jeong and Efferth, Thomas. (2017) Antileukemic ancistrobenomine B and related 5,1'-coupled naphthylisoquinoline alkaloids from the Chinese liana Ancistrocladus tectorius. Fitoterapia, 121. pp. 76-85.

Tshitenge, Dieudonné Tshitenge and Feineis, Doris and Mudogo, Virima and Kaiser, Marcel and Brun, Reto and Bringmann, Gerhard. (2017) Antiplasmodial ealapasamines A-C,'mixed' naphthylisoquinoline dimers from the Central African liana Ancistrocladus ealaensis. Scientific Reports, 7. p. 5767.

De Mieri, Maria and Monteleone, Giannicola and Ismajili, Isidor and Kaiser, Marcel and Hamburger, Matthias. (2017) Antiprotozoal activity-based profiling of a dichloromethane extract from anthemis nobilis flowers. Journal of Natural Products, 80 (2). pp. 459-470.

Chianese, Giuseppina and Silber, Johanna and Luciano, Paolo and Merten, Christian and Erpenbeck, Dirk and Topaloglu, Bülent and Kaiser, Marcel and Tasdemir, Deniz. (2017) Antiprotozoal linear furanosesterterpenoids from the marine sponge Ircinia oros. Journal of natural products, 80 (9). pp. 2566-2571.

Smyrniotopoulos, Vangelis and Merten, Christian and Kaiser, Marcel and Tasdemir, Deniz. (2017) Bifurcatriol, a new antiprotozoal acyclic diterpene from the brown alga Bifurcaria bifurcata. Marine drugs, 15 (8). p. 245.

Bode, Edna and He, Yue and Vo, Tien Duy and Schultz, Roland and Kaiser, Marcel and Bode, Helge B.. (2017) Biosynthesis and function of simple amides in Xenorhabdus doucetiae. Environmental Microbiology, 19 (11). pp. 4564-4575.

Cai, Xiaofeng and Challinor, Victoria L. and Zhao, Lei and Reimer, Daniela and Adihou, Hélène and Grün, Peter and Kaiser, Marcel and Bode, Helge B.. (2017) Biosynthesis of the antibiotic nematophin and its elongated derivatives in entomopathogenic bacteria. Organic letters, 19 (4). pp. 806-809.

Li, Jun and Seupel, Raina and Feineis, Doris and Mudogo, Virima and Kaiser, Marcel and Brun, Reto and Brünnert, Daniela and Chatterjee, Manik and Seo, Ean-Jeong and Efferth, Thomas and Bringmann, Gerhard. (2017) Dioncophyllines C2, D2, and F and related naphthylisoquinoline alkaloids from the congolese liana Ancistrocladus ileboensis with potent activities against Plasmodium falciparum and against multiple myeloma and leukemia cell lines. Journal of natural products, 80 (2). pp. 443-458.

Cai, Xiaofeng and Nowak, Sarah and Wesche, Frank and Bischoff, Iris and Kaiser, Marcel and Fürst, Robert and Bode, Helge B.. (2017) Entomopathogenic bacteria use multiple mechanisms for bioactive peptide library design. Nature Chemistry, 9 (4). pp. 379-386.

Steiniger, Charlotte and Hoffmann, Sylvester and Mainz, Andi and Kaiser, Marcel and Voigt, Kerstin and Meyer, Vera and Süssmuth, Roderich D.. (2017) Harnessing fungal nonribosomal cyclodepsipeptide synthetases for mechanistic insights and tailored engineering. Chemical Science, 8 (11). pp. 7834-7843.

Tallini, Luciana R. and Osorio, Edison H. and Santos, Vanessa Dias Dos and Borges, Warley de Souza and Kaiser, Marcel and Viladomat, Francesc and Zuanazzi, José Angelo S. and Bastida, Jaume. (2017) Hippeastrum reticulatum (Amaryllidaceae): alkaloid profiling, biological activities and molecular docking. Molecules, 22 (12). E2191.

Li, Jun and Seupel, Raina and Bruhn, Torsten and Feineis, Doris and Kaiser, Marcel and Brun, Reto and Mudogo, Virima and Awale, Suresh and Bringmann, Gerhard. (2017) Jozilebomines A and B, naphthylisoquinoline dimers from the congolese liana ancistrocladus ileboensis, with antiausterity activities against the PANC-1 human pancreatic cancer cell line. Journal of natural products, 80 (10). pp. 2807-2817.

Pagliero, Romina J. and Kaiser, Marcel and Brun, Reto and Nieto, Marcelo J. and Mazzieri, María R.. (2017) Lead selection of antiparasitic compounds from a focused library of benzenesulfonyl derivatives of heterocycles. Bioorganic & medicinal chemistry, 27 (17). pp. 3945-3949.

Bruno, Stefano and Uliassi, Elisa and Zaffagnini, Mirko and Prati, Federica and Bergamini, Christian and Amorati, Riccardo and Paredi, Gianluca and Margiotta, Marilena and Conti, Paola and Costi, Maria Paola and Kaiser, Marcel and Cavalli, Andrea and Fato, Romana and Bolognesi, Maria Laura. (2017) Molecular basis for covalent inhibition of glyceraldehyde-3-phosphate dehydrogenase by a 2-phenoxy-1,4-naphthoquinone small molecule. Chemical Biology and Drug Design, 90 (2). pp. 225-235.

Faist, Johanna and Hinteregger, Clemens and Seebacher, Werner and Saf, Robert and Mäser, Pascal and Kaiser, Marcel and Weis, Robert. (2017) New derivatives of 7-chloroquinolin-4-amine with antiprotozoal activity. Bioorganic & medicinal chemistry, 25 (3). pp. 941-948.

Hochegger, Patrick and Faist, Johanna and Seebacher, Werner and Saf, Robert and Mäser, Pascal and Kaiser, Marcel and Weis, Robert. (2017) New derivatives of quinoline-4-carboxylic acid with antiplasmodial activity. Bioorganic & medicinal chemistry, 25 (7). pp. 2251-2259.

Nnadi, Charles Okeke and Nwodo, Ngozi Justina and Kaiser, Marcel and Brun, Reto and Schmidt, Thomas J.. (2017) Steroid Alkaloids from Holarrhena africana with Strong Activity against Trypanosoma brucei rhodesiense. Molecules, 22 (7). E1129.

Cai, Xiaofeng and Shi, Yi-Ming and Pöhlmann, Nicole and Revermann, Ole and Bahner, Isabel and Pidot, Sacha J. and Wesche, Frank and Lackner, Helmut and Büchel, Claudia and Kaiser, Marcel and Richter, Christian and Schwalbe, Harald and Stinear, Timothy P. and Zeeck, Axel and Bode, Helge B.. (2017) Structure and biosynthesis of isatropolones, bioactive amine-scavenging fluorescent natural products from streptomyces Go66. Angewandte Chemie International Edition, 56 (18). pp. 4945-4949.

Cadelis, Melissa M. and Bourguet-Kondracki, Marie-Lise and Dubois, Joëlle and Kaiser, Marcel and Brunel, Jean Michel and Barker, David and Copp, Brent R.. (2017) Structure-activity relationship studies on thiaplidiaquinones A and B as novel inhibitors of Plasmodium falciparum and farnesyltransferase. Bioorganic & medicinal chemistry, 25 (16). pp. 4433-4443.

Tran, Huu-Anh and Zheng, Zhaoyan and Wen, Xianghui and Manivannan, Srinivasan and Pastor, Arnaud and Kaiser, Marcel and Brun, Reto and Snyder, Floyd F. and Back, Thomas G.. (2017) Synthesis and activity of nucleoside-based antiprotozoan compounds. Bioorganic & medicinal chemistry, 25 (7). pp. 2091-2104.

Pearce, A. Norrie and Kaiser, Marcel and Copp, Brent R.. (2017) Synthesis and antimalarial evaluation of artesunate-polyamine and trioxolane-polyamine conjugates. European journal of medicinal chemistry, 140. pp. 595-603.

Mohsin, Noor-Ul-Amin and Seebacher, Werner and Faist, Johanna and Hochegger, Patrick and Kaiser, Marcel and Mäser, Pascal and Belaj, Ferdinand and Saf, Robert and Kretschmer, Nadine and Alajlani, Muaaz and Turek, Ivana and Brantner, Adelheid and Bauer, Rudolf and Bucar, Franz and Weis, Robert. (2017) Synthesis of new 1-benzyl tetrahydropyridinylidene ammonium salts and their antimicrobial and anticellular activities. European journal of medicinal chemistry, 143. pp. 97-106.

Greve, Hippolyt L. and Kaiser, Marcel and Brun, Reto and Schmidt, Thomas J.. (2017) Terpenoids from the oleo-gum-resin of Boswellia serrata and their antiplasmodial effects In Vitro. Planta medica, 83 (14-15). pp. 1214-1226.

Papadopoulou, Maria V. and Bloomer, William D. and Rosenzweig, Howard S. and Kaiser, Marcel. (2017) The antitrypanosomal and antitubercular activity of some nitro(triazole/imidazole)-based aromatic amines. European Journal of Medicinal Chemistry, 138. pp. 1106-1113.

2016

Silveira, Narjara and Saar, Julia and Santos, Alan Diego C. and Barison, Andersson and Sandjo, Louis P. and Kaiser, Marcel and Schmidt, Thomas J. and Biavatti, Maique W.. (2016) A new alkamide with an endoperoxide structure from acmella ciliata (asteraceae) and its in vitro antiplasmodial activity. Molecules, 21 (6). pp. 1-10.

Pirttimaa, Minni and Nasereddin, Abedelmajeed and Kopelyanskiy, Dmitry and Kaiser, Marcel and Yli-Kauhaluoma, Jari and Oksman-Caldentey, Kirsi-Marja and Brun, Reto and Jaffe, Charles L. and Moreira, Vânia M. and Alakurtti, Sami. (2016) Abietane-type diterpenoid amides with highly potent and selective activity against Leishmania donovani and Trypanosoma cruzi. Journal of natural products, 79 (2). pp. 362-368.

Bringmann, Gerhard and Seupel, Raina and Feineis, Doris and Zhang, Guoliang and Xu, Minjuan and Wu, Jun and Kaiser, Marcel and Brun, Reto and Seo, Ean-Jeong and Efferth, Thomas. (2016) Ancistectorine D, a naphthylisoquinoline alkaloid with antiprotozoal and antileukemic activities, and further 5,8'- and 7,1'-linked metabolites from the Chinese liana Ancistrocladus tectorius. Fitoterapia, 115. pp. 1-8.

Faist, Johanna and Seebacher, Werner and Saf, Robert and Brun, Reto and Kaiser, Marcel and Weis, Robert. (2016) Antiprotozoal activity of bicycles featuring a dimethylamino group at their bridgehead. Bioorganic & medicinal chemistry, 24 (16). pp. 3781-3789.

Papadopoulou, Maria V. and Bloomer, William D. and Rosenzweig, Howard S. and Wilkinson, Shane R. and Szular, Joanna and Kaiser, Marcel. (2016) Antitrypanosomal activity of 5-nitro-2-aminothiazole-based compounds. European journal of medicinal chemistry, 117. pp. 179-186.

Cal, Monica and Ioset, Jean-Robert and Fügi, Matthia A. and Mäser, Pascal and Kaiser, Marcel. (2016) Assessing anti-T. cruzi candidates in vitro for sterile cidality. International journal for parasitology. Drugs and drug resistance, 6 (3). pp. 165-170.

Seupel, Raina and Hertlein-Amslinger, Barbara and Gulder, Tanja and Stawski, Philipp and Kaiser, Marcel and Brun, Reto and Bringmann, Gerhard. (2016) Directed synthesis of all four pure stereoisomers of the N,C-Coupled naphthylisoquinoline alkaloid ancistrocladinium A. Organic letters, 18 (24). pp. 6508-6511.

Nogueira, Mauro S. and Da Costa, Fernando B. and Brun, Reto and Kaiser, Marcel and Schmidt, Thomas J.. (2016) Ent-pimarane and ent-kaurane diterpenes from Aldama discolor (asteraceae) and their antiprotozoal activity. Molecules, 21 (9). p. 1237.

Atay, Irem and Kirmizibekmez, Hasan and Kaiser, Marcel and Akaydin, Galip and Yesilada, Erdem and Tasdemir, Deniz. (2016) Evaluation of in vitro antiprotozoal activity of Ajuga laxmannii and its secondary metabolites. Pharmaceutical biology, 54 (9). pp. 1808-1814.

Russell, Stephanie and Rahmani, Raphaël and Jones, Amy J. and Newson, Harriet L. and Neilde, Kevin and Cotillo, Ignacio and Rahmani Khajouei, Marzieh and Ferrins, Lori and Qureishi, Sana and Nguyen, Nghi and Martinez-Martinez, Maria S. and Weaver, Donald F. and Kaiser, Marcel and Riley, Jennifer and Thomas, John and De Rycker, Manu and Read, Kevin D. and Flematti, Gavin R. and Ryan, Eileen and Tanghe, Scott and Rodriguez, Ana and Charman, Susan A. and Kessler, Albane and Avery, Vicky M. and Baell, Jonathan B. and Piggott, Matthew J.. (2016) Hit-to-lead optimization of a novel class of potent, broad-spectrum trypanosomacides. Journal of Medicinal Chemistry, 59 (21). pp. 9686-9720.

Papadopoulou, Maria V. and Bloomer, William D. and Rosenzweig, Howard S. and Wilkinson, Shane R. and Szular, Joanna and Kaiser, Marcel. (2016) Nitrotriazole-based acetamides and propanamides with broad spectrum antitrypanosomal activity. European journal of medicinal chemistry, 123. pp. 895-904.

Zheng, Zhaoyan and Tran, Huu-Anh and Manivannan, Srinivasan and Wen, Xianghui and Kaiser, Marcel and Brun, Reto and Snyder, Floyd F. and Back, Thomas G.. (2016) Novel nucleoside-based antimalarial compounds. Bioorganic & medicinal chemistry letters, 26 (12). pp. 2861-2865.

Kedzierska, Ewa and Orzelska, Jolanta and Perković, Ivana and Knežević, Danijel and Fidecka, Sylwia and Kaiser, Marcel and Zorc, Branka. (2016) Pharmacological effects of primaquine ureas and semicarbazides on the central nervous system in mice and antimalarial activity in vitro. Fundamental and clinical pharmacology, 30. pp. 58-69.

Hiltensperger, Georg and Hecht, Nina and Kaiser, Marcel and Rybak, Jens-Christoph and Hoerst, Alexander and Dannenbauer, Nicole and Müller-Buschbaum, Klaus and Bruhn, Heike and Esch, Harald and Lehmann, Leane and Meinel, Lorenz and Holzgrabe, Ulrike. (2016) Quinolone amides as anti-trypanosomal lead compounds with in vivo activity. Antimicrobial agents and chemotherapy, 60 (8). pp. 4442-4452.

Karaaslan, Cigdem and Kaiser, Marcel and Brun, Reto and Göker, Hakan. (2016) Synthesis and potent antiprotozoal activity of mono/di amidino 2-anilinobenz-imidazoles versus Plasmodium falciparum and Trypanosoma brucei rhodesiense. Bioorganic and Medicinal Chemistry, 24 (18). pp. 4038-4044.

Ahmad, Sarfraz and Seebacher, Werner and Faist, Johanna and Kaiser, Marcel and Brun, Reto and Saf, Robert and Weis, Robert. (2016) The antiprotozoal potencies of newly prepared 3-azabicyclo[3.2.2]nonanes. Archives of pharmacal research, 39 (10). pp. 1391-1403.

Houël, Emeline and Nardella, Flore and Jullian, Valérie and Valentin, Alexis and Vonthron-Sénécheau, Catherine and Villa, Pascal and Obrecht, Adeline and Kaiser, Marcel and Bourreau, Eliane and Odonne, Guillaume and Fleury, Marie and Bourdy, Geneviève and Eparvier, Véronique and Deharo, Eric and Stien, Didier. (2016) Wayanin and guaijaverin, two active metabolites found in a Psidium acutangulum mart. ex DC (syn. P. persoonii McVaugh) (Myrtaceae) antimalarial decoction from the Wayana Amerindians. Journal of ethnopharmacology, 187. pp. 241-248.

2015

Prati, Federica and Bergamini, Christian and Molina, Maria Teresa and Falchi, Federico and Cavalli, Andrea and Kaiser, Marcel and Brun, Reto and Fato, Romana and Bolognesi, Maria Laura. (2015) 2-Phenoxy-1,4-naphthoquinones : from a multitarget antitrypanosomal to a potential antitumor profile. Journal of medicinal chemistry, 58 (16). pp. 6422-6434.

Papadopoulou, Maria V. and Bloomer, William D. and Rosenzweig, Howard S. and O'Shea, Ivan P. and Wilkinson, Shane R. and Kaiser, Marcel. (2015) 3-Nitrotriazole-based piperazides as potent antitrypanosomal agents. European journal of medicinal chemistry, 103. pp. 325-334.

Rahmani, Raphaël and Ban, Kung and Jones, Amy J. and Ferrins, Lori and Ganame, Danny and Sykes, Melissa L. and Avery, Vicky M. and White, Karen L. and Ryan, Eileen and Kaiser, Marcel and Charman, Susan A. and Baell, Jonathan B.. (2015) 6-Arylpyrazine-2-carboxamides : a new core for Trypanosoma brucei inhibitors. Journal of medicinal chemistry, 58 (17). pp. 6753-6765.

Ríos Martínez, Carlos H. and Miller, Florence and Ganeshamoorthy, Kayathiri and Glacial, Fabienne and Kaiser, Marcel and de Koning, Harry P. and Eze, Anthonius A. and Lagartera, Laura and Herraiz, Tomás and Dardonville, Christophe. (2015) A new nonpolar n-hydroxy imidazoline lead compound with improved activity in a murine model of late-stage Trypanosoma brucei brucei infection is not cross-resistant with diamidines. Antimicrobial agents and chemotherapy, Vol. 59, H. 2. pp. 890-904.

Nollmann, Friederike I. and Heinrich, Antje K. and Brachmann, Alexander O. and Morisseau, Christophe and Mukherjee, Krishnendu and Casanova-Torres, Ángel M. and Strobl, Frederic and Kleinhans, David and Kinski, Sebastian and Schultz, Katharina and Beeton, Michael L. and Kaiser, Marcel and Chu, Ya-Yun and Phan Ke, Long and Thanwisai, Aunchalee and Bozhüyük, Kenan A. J. and Chantratita, Narisara and Götz, Friedrich and Waterfield, Nick R. and Vilcinskas, Andreas and Stelzer, Ernst H. K. and Goodrich-Blair, Heidi and Hammock, Bruce D. and Bode, Helge B.. (2015) A photorhabdus natural product inhibits insect juvenile hormone epoxide hydrolase. ChemBioChem, Vol. 16, H. 5. pp. 766-771.

Inahashi, Yuki and Iwatsuki, Masato and Ishiyama, Aki and Matsumoto, Atsuko and Hirose, Tomoyasu and Oshita, Jun and Sunazuka, Toshiaki and Panbangred, Watanalai and Takahashi, Yoko and Kaiser, Marcel and Otoguro, Kazuhiko and O̅mura, Satoshi. (2015) Actinoallolides A-E, new anti-trypanosomal macrolides, produced by an endophytic actinomycete, actinoallomurus fulvus MK10-036. Organic letters, Vol. 17, H. 4. pp. 864-867.

Thao, Nguyen Phuong and Luyen, Bui Thi Thuy and Brun, Reto and Kaiser, Marcel and Van Kiem, Phan and Van Minh, Chau and Schmidt, Thomas J. and Kang, Jong Seong and Kim, Young Ho. (2015) Anti-protozoal activities of cembrane-type diterpenes from Vietnamese soft corals. Molecules, Vol. 20, H. 7. pp. 12459-12468.

Montalvo-Quirós, Sandra and Taladriz-Sender, Andrea and Kaiser, Marcel and Dardonville, Christophe. (2015) Antiprotozoal activity and DNA binding of dicationic acridones. Journal of medicinal chemistry, 58 (4). pp. 1940-1949.

Kaiser, Marcel and Mäser, Pascal and Tadoori, Leela Pavan and Ioset, Jean-Robert and Brun, Reto. (2015) Antiprotozoal activity profiling of approved drugs : a starting point toward drug repositioning. PLoS ONE, Vol. 10, H. 8 , e0135556.

Cretton, Sylvian and Bréant, Lise and Pourrez, Lucie and Ambuehl, Chiara and Perozzo, Remo and Marcourt, Laurence and Kaiser, Marcel and Cuendet, Muriel and Christen, Philippe. (2015) Chemical constituents from Waltheria indica exert in vitro activity against Trypanosoma brucei and T. cruzi. Fitoterapia, 105. pp. 55-60.

Royo, Santiago and Rodríguez, Santiago and Schirmeister, Tanja and Kesselring, Jochen and Kaiser, Marcel and González, Florenci V.. (2015) Dipeptidyl enoates as potent rhodesain inhibitors that display a dual mode of action. ChemMedChem, 10 (9). pp. 1484-1487.

Mital, Alka and Murugesan, Dinakaran and Kaiser, Marcel and Yeates, Clive and Gilbert, Ian H.. (2015) Discovery and optimisation studies of antimalarial phenotypic hits. European journal of medicinal chemistry, 103. pp. 530-538.

Woodland, Andrew and Thompson, Stephen and Cleghorn, Laura A. T. and Norcross, Neil and De Rycker, Manu and Grimaldi, Raffaella and Hallyburton, Irene and Rao, Bhavya and Norval, Suzanne and Stojanovski, Laste and Brun, Reto and Kaiser, Marcel and Frearson, Julie A. and Gray, David W. and Wyatt, Paul G. and Read, Kevin D. and Gilbert, Ian H.. (2015) Discovery of inhibitors of Trypanosoma brucei by phenotypic screening of a focused protein kinase library. ChemMedChem, 10 (11). pp. 1809-1820.

Papadopoulou, Maria V. and Bloomer, William D. and Rosenzweig, Howard S. and O'Shea, Ivan P. and Wilkinson, Shane R. and Kaiser, Marcel and Chatelain, Eric and Ioset, Jean-Robert. (2015) Discovery of potent nitrotriazole-based antitrypanosomal agents : in vitro and in vivo evaluation. Bioorganic & medicinal chemistry, 23 (19). pp. 6467-6476.

Cheikh-Ali, Zakaria and Glynou, Kyriaki and Ali, Tahir and Ploch, Sebastian and Kaiser, Marcel and Thines, Marco and Bode, Helge B. and Maciá-Vicente, Jose G.. (2015) Diversity of exophillic acid derivatives in strains of an endophytic Exophiala sp. Phytochemistry : an international journal of plant biochemistry, 118. pp. 83-93.

Nwodo, Ngozi and Okoye, Festus and Lai, Daowan and Debbab, Abdesammed and Kaiser, Marcel and Brun, Reto and Proksch, Peter. (2015) Evaluation of the in vitro trypanocidal activity of methylated flavonoid constituents of Vitex simplicifolia leaves. BMC complementary and alternative medicine, Vol. 15 , 82.

Hemberger, Yasmin and Zhang, Guoliang and Brun, Reto and Kaiser, Marcel and Bringmann, Gerhard. (2015) Highly antiplasmodial non-natural oxidative products of dioncophylline A: synthesis, absolute configuration, and conformational stability. Chemistry, a European journal, 21 (41). pp. 14507-14518.

Jones, Amy J. and Kaiser, Marcel and Avery, Vicky M.. (2015) Identification and characterization of FTY720 for the treatment of human African trypanosomiasis. Antimicrobial agents and chemotherapy, 60 (3). pp. 1859-1861.

Herrmann, Fabian C. and Lenz, Mairin and Jose, Joachim and Kaiser, Marcel and Brun, Reto and Schmidt, Thomas J.. (2015) In silico identification and in vitro activity of novel natural inhibitors of Trypanosoma brucei glyceraldehyde-3-phosphate-dehydrogenase. Molecules, Vol. 20, H. 9. pp. 16154-16169.

Nollmann, Friederike I. and Dauth, Christina and Mulley, Geraldine and Kegler, Carsten and Kaiser, Marcel and Waterfield, Nick R. and Bode, Helge B.. (2015) Insect-specific production of new GameXPeptides in Photorhabdus luminescens TTO1, widespread natural products in entomopathogenic bacteria. ChemBioChem : a European journal of chemical biology, Vol. 16, H. 2. pp. 205-208.

Keller, Lena and Plaza, Alberto and Dubiella, Christian and Groll, Michael and Kaiser, Marcel and Müller, Rolf. (2015) Macyranones : structure, biosynthesis, and binding mode of an unprecedented epoxyketone that targets the 20S proteasome. The journal of the American Chemical Society, Vol. 137, H. 25. pp. 8121-8130.

Papadopoulou, Maria V. and Bloomer, William D. and Lepesheva, Galina I. and Rosenzweig, Howard S. and Kaiser, Marcel and Aguilera-Venegas, Benjamín and Wilkinson, Shane R. and Chatelain, Eric and Ioset, Jean-Robert. (2015) Novel 3-nitrotriazole-based amides and carbinols as bifunctional antichagasic agents. Journal of medicinal chemistry, 58 (3). pp. 1307-1319.

Ellendorff, Therese and Brun, Reto and Kaiser, Marcel and Sendker, Jandirk and Schmidt, Thomas J.. (2015) PLS-prediction and confirmation of hydrojuglone glucoside as the antitrypanosomal constituent of "Juglans spp.". Molecules, Vol. 20, H. 6. pp. 10082-10094.

Daeppen, Christophe and Kaiser, Marcel and Neuburger, Markus and Gademann, Karl. (2015) Preparation of antimalarial endoperoxides by a formal [2 + 2 + 2] cycloaddition. Organic letters, 17 (21). pp. 5420-5423.

Kaiser, Marcel and Maes, Louis and Tadoori, Leela Pavan and Spangenberg, Thomas and Ioset, Jean-Robert. (2015) Repurposing of the open access malaria box for kinetoplastid diseases identifies novel active scaffolds against trypanosomatids. Journal of biomolecular screening, Vol. 20, H. 5. pp. 634-645.

Montesino, Núria Llurba and Kaiser, Marcel and Brun, Reto and Schmidt, Thomas J.. (2015) Search for antiprotozoal activity in herbal medicinal preparations : new natural leads against neglected tropical diseases. Molecules, Vol. 20, H. 8. pp. 14118-14138.

Bode, Edna and Brachmann, Alexander O. and Kegler, Carsten and Simsek, Rukayye and Dauth, Christina and Zhou, Qiuqin and Kaiser, Marcel and Klemmt, Petra and Bode, Helge B.. (2015) Simple "on-demand" production of bioactive natural products. ChemBioChem, Vol. 16, H. 7. pp. 1115-1119.

Bode, Helge B. and Brachmann, Alexander O. and Jadhav, Kirtikumar B. and Seyfarth, Lydia and Dauth, Christina and Fuchs, Sebastian W. and Kaiser, Marcel and Waterfield, Nick R. and Sack, Holger and Heinemann, Stefan H. and Arndt, Hans-Dieter. (2015) Structure elucidation and activity of kolossin A, the D-/L-Pentadecapeptide product of a giant nonribosomal peptide synthetase. Angewandte Chemie, Jg. 54, Nr. 35. pp. 10352-10355.

Ahmad, Sarfraz and Seebacher, Werner and Wolkinger, Volker and Presser, Armin and Faist, Johanna and Kaiser, Marcel and Brun, Reto and Saf, Robert and Weis, Robert. (2015) Synthesis and antiprotozoal activities of new 3-azabicyclo[3.2.2]nonanes. Archives of pharmacal research, Vol. 38, H. 8. pp. 1455-1467.

Seebacher, Werner and Wolkinger, Volker and Faist, Johanna and Kaiser, Marcel and Brun, Reto and Saf, Robert and Bucar, Franz and Gröblacher, Barbara and Brantner, Adelheid and Merino, Virginia and Kalia, Yogeshvar and Scapozza, Leonardo and Perozzo, Remo and Weis, Robert. (2015) Synthesis of 3-azabicyclo[3.2.2]nonanes and their antiprotozoal activities. Bioorganic & medicinal chemistry letters, Vol. 25, H. 7. pp. 1390-1393.

Rodenko, Boris and Wanner, Martin J. and Alkhaldi, Abdulsalam A. M. and Ebiloma, Godwin U. and Barnes, Rebecca L. and Kaiser, Marcel and Brun, Reto and McCulloch, Richard and Koomen, Gerrit-Jan and de Koning, Harry P.. (2015) Targeting the parasite's DNA with methyltriazenyl purine analogs is a safe, selective, and efficacious antitrypanosomal strategy. Antimicrobial agents and chemotherapy, 59 (11). pp. 6708-6716.

2014

de Meijere, Armin and Kozhushkov, Sergei I. and Yufit, Dmitrii S. and Grosse, Christian and Kaiser, Marcel and Raev, Vitaly A.. (2014) (2R,1'S,2'R)- and (2S,1'S,2'R)-3-[2-Mono(di,tri)fluoromethylcyclopropyl]alanines and their incorporation into hormaomycin analogues. Beilstein journal of organic chemistry, Vol. 10. pp. 2844-2857.

Wube, Abraham and Hüfner, Antje and Seebacher, Werner and Kaiser, Marcel and Brun, Reto and Bauer, Rudolf and Bucar, Franz. (2014) 1,2-substituted 4-(1H)-quinolones : synthesis, antimalarial and antitrypanosomal activities in vitro. Molecules, Vol. 19, H. 9. pp. 14204-14220.

Carballeira, Néstor M. and Bwalya, Angela Gono and Itoe, Maurice Ayamba and Andricopulo, Adriano D. and Cordero-Maldonado, María Lorena and Kaiser, Marcel and Mota, Maria M. and Crawford, Alexander D. and Guido, Rafael V. C. and Tasdemir, Deniz. (2014) 2-Octadecynoic acid as a dual life stage inhibitor of Plasmodium infections and plasmodial FAS-II enzymes. Bioorganic & medicinal chemistry letters, Vol. 24, H. 17. pp. 4151-4157.

Dong, Yuxiang and Wang, Xiaofang and Cal, Monica and Kaiser, Marcel and Vennerstrom, Jonathan L.. (2014) Activity of diimidazoline amides against African trypanosomiasis. Bioorganic & medicinal chemistry letters, Vol. 24, H. 3. pp. 944-948.

Mokoka, Tsholofelo A. and Peter, Xolani K. and Fouche, Gerda and Moodley, Nivan and Adams, Michael and Hamburger, Matthias and Kaiser, Marcel and Brun, Reto and Maharaj, Vinesh and Koorbanally, Neil. (2014) Antileishmanial activity of 12-methoxycarnosic acid from Salvia repens Buch. ex Benth. (Lamiaceae). South African journal of botany, Vol. 90. pp. 93-95.

Grundmann, Florian and Kaiser, Marcel and Schiell, Matthias and Batzer, Andreas and Kurz, Michael and Thanwisai, Aunchalee and Chantratita, Narisara and Bode, Helge B.. (2014) Antiparasitic chaiyaphumines from Entomopathogenic xenorhabdus sp. PB61.4. Journal of natural products, Vol. 77, H. 4. pp. 779-783.

Ríos Martínez, Carlos H. and Lagartera, Laura and Kaiser, Marcel and Dardonville, Christophe. (2014) Antiprotozoal activity and DNA binding of N-substituted N-phenylbenzamide and 1,3-diphenylurea bisguanidines. European journal of medicinal chemistry, 81. pp. 481-491.

Orhan, Ilkay Erdogan and Sener, Bilge and Kaiser, Marcel and Brun, Reto and Tasdemir, Deniz. (2014) Antiprotozoal activity and cytotoxicity of Lycopodium clavatum and Lycopodium complanatum subsp. chamaecyparissus extracts. Turkish journal of biochemistry, Vol. 38, H. 4. pp. 403-408.

Carvalho, Samir Aquino and Kaiser, Marcel and Brun, Reto and Silva, Edson Ferreira da and Fraga, Carlos Alberto Manssour. (2014) Antiprotozoal activity of (e)-cinnamic N-acylhydrazone derivatives. Molecules, Vol. 19, H. 12. pp. 20374-20381.

Althaus, Julia B. and Jerz, Gerold and Winterhalter, Peter and Kaiser, Marcel and Brun, Reto and Schmidt, Thomas J.. (2014) Antiprotozoal activity of Buxus sempervirens and activity-guided isolation of O-tigloylcyclovirobuxeine-B as the main constituent active against Plasmodium falciparum. Molecules : a journal of synthetic chemistry and natural product chemistry, Vol. 19, H. 5. pp. 6184-6201.

Althaus, Julia B. and Kaiser, Marcel and Brun, Reto and Schmidt, Thomas J.. (2014) Antiprotozoal activity of achillea ptarmica (Asteraceae) and its main alkamide constituents. Molecules : a journal of synthetic chemistry and natural product chemistry, Vol. 19, H. 5. pp. 6428-6438.

Hata, Yoshie and Ebrahimi, Samad Nejad and De Mieri, Maria and Zimmermann, Stefanie and Mokoka, Tsholofelo and Naidoo, Dashnie and Fouche, Gerda and Maharaj, Vinesh and Kaiser, Marcel and Brun, Reto and Potterat, Olivier and Hamburger, Matthias. (2014) Antitrypanosomal isoflavan quinones from Abrus precatorius. Fitoterapia, Vol. 93. pp. 81-87.

Ayyari, Mahdi and Salehi, Peyman and Ebrahimi, Samad Nejad and Zimmermann, Stefanie and Portmann, Lena and Krauth-Siegel, R. Luise and Kaiser, Marcel and Brun, Reto and Rezadoost, Hassan and Rezazadeh, Shamsali and Hamburger, Matthias. (2014) Antitrypanosomal isothiocyanate and thiocarbamate glycosides from Moringa peregrina. Planta Medica, 80 (1). pp. 86-89.

Cretton, Sylvian and Breant, Lise and Pourrez, Lucie and Ambuehl, Chiara and Marcourt, Laurence and Ebrahimi, Samad Nejad and Hamburger, Matthias and Perozzo, Remo and Karimou, Soumana and Kaiser, Marcel and Cuendet, Muriel and Christen, Philippe. (2014) Antitrypanosomal quinoline alkaloids from the roots of Waltheria indica. Journal of natural products, Vol. 77, H. 10. pp. 2304-2311.

Usuki, Toyonobu and Sato, Makiko and Hara, Shihori and Yoshimoto, Yukiko and Kondo, Ryosuke and Zimmermann, Stefanie and Kaiser, Marcel and Brun, Reto and Hamburger, Matthias and Adams, Michael. (2014) Antitrypanosomal structure-activity-relationship study of synthetic cynaropicrin derivatives. Bioorganic & medicinal chemistry letters, Vol. 24, H. 3. pp. 794-798.

Portmann, Cyril and Sieber, Simon and Wirthensohn, Silvan and Blom, Judith F. and Da Silva, Laeticia and Baudat, Emilie and Kaiser, Marcel and Brun, Reto and Gademann, Karl. (2014) Balgacyclamides, antiplasmodial heterocyclic peptides from Microcystis aeruguinosa EAWAG 251. Journal of natural products, Vol. 77, H. 3. pp. 557-562.

Persch, Elke and Bryson, Steve and Todoroff, Nickolay K. and Eberle, Christian and Thelemann, Jonas and Dirdjaja, Natalie and Kaiser, Marcel and Weber, Maria and Derbani, Hassan and Brun, Reto and Schneider, Gisbert and Pai, Emil F. and Krauth-Siegel, R. Luise and Diederich, François. (2014) Binding to large enzyme pockets : small-molecule inhibitors of trypanothione reductase. ChemMedChem, Vol. 9, H. 8. pp. 1880-1891.

Kronenwerth, Max and Brachmann, Alexander O. and Kaiser, Marcel and Bode, Helge B.. (2014) Bioactive derivatives of isopropylstilbene from mutasynthesis and chemical synthesis. ChemBioChem : a European journal of chemical biology, Vol. 15, H. 18. pp. 2689-2691.

Kronenwerth, Max and Bozhüyük, Kenan A. J. and Kahnt, Astrid S. and Steinhilber, Dieter and Gaudriault, Sophie and Kaiser, Marcel and Bode, Helge B.. (2014) Characterisation of taxlllaids A-G : natural products from Xenorhabdus indica. Chemistry : a European journal, Vol. 20, H. 52. pp. 17478-17487.

Giordani, Federica and Buschini, Annamaria and Baliani, Alessandro and Kaiser, Marcel and Brun, Reto and Barrett, Michael P. and Pellacani, Claudia and Poli, Paola and Gilbert, Ian H.. (2014) Characterization of a melamino nitroheterocycle as a potential lead for the treatment of human african trypanosomiasis. Antimicrobial agents and chemotherapy, Vol. 58, H. 10. pp. 5747-5757.

Fuchs, Sebastian W. and Grundmann, Florian and Kurz, Michael and Kaiser, Marcel and Bode, Helge B.. (2014) Fabclavines : bioactive peptide-polyketide-polyamino hybrids from Xenorhabdus. ChemBioChem : a European journal of chemical biology, Vol. 15, H. 4. pp. 512-516.

Julianti, Tasqiah and De Mieri, Maria and Zimmermann, Stefanie and Ebrahimi, Samad N. and Kaiser, Marcel and Neuburger, Markus and Raith, Melanie and Brun, Reto and Hamburger, Matthias. (2014) HPLC-based activity profiling for antiplasmodial compounds in the traditional Indonesian medicinal plant Carica papaya L. Journal of ethnopharmacology, Vol. 155, H. 1. pp. 426-434.

Schmidt, Thomas J. and Da Costa, Fernando B. and Lopes, Norberto P. and Kaiser, Marcel and Brun, Reto. (2014) In Silico prediction and experimental evaluation of furanoheliangolide sesquiterpene lactones as potent agents against Trypanosoma brucei rhodesiense. Antimicrobial agents and chemotherapy, Vol. 58, H. 1. pp. 325-332.

Bapela, M. Johanna and Meyer, J. J. Marion and Kaiser, Marcel. (2014) In vitro antiplasmodial screening of ethnopharmacologically selected South African plant species used for the treatment of malaria. Journal of ethnopharmacology : an interdisciplinary journal devoted to bioscientific research on indigenous drugs, Vol. 156. pp. 370-373.

Harms, Henrik and Rempel, Viktor and Kehraus, Stefan and Kaiser, Marcel and Hufendiek, Peter and Müller, Christa E. and König, Gabriele M.. (2014) Indoloditerpenes from a marine-derived fungal strain of Dichotomomyces cejpii with antagonistic activity at GPR18 and cannabinoid receptors. Journal of natural products, Vol. 77, H. 3. pp. 673-677.

Wang, Jiayi and Kaiser, Marcel and Copp, Brent R.. (2014) Investigation of indolglyoxamide and indolacetamide analogues of polyamines as antimalarial and antitrypanosomal agents. Marine drugs, Vol. 12, H. 6. pp. 3138-3160.

Fügi, Matthias A. and Kaiser, Marcel and Tanner, Marcel and Schneiter, Roger and Mäser, Pascal and Guan, Xue Li. (2014) Match-making for posaconazole through systems thinking. Trends in parasitology, Vol. 31, H. 2. pp. 46-51.

Kaiser, Marcel. New drugs against trypanosomatid parasites : rediscovery of fexinidazole. 2014, Doctoral Thesis, University of Basel, Faculty of Science.

Papadopoulou, Maria V. and Bloomer, William D. and Rosenzweig, Howard S. and Wilkinson, Shane R. and Kaiser, Marcel. (2014) Novel nitro(triazole/imidazole)-based heteroarylamides/sulfonamides as potential antitrypanosomal agents. European journal of medicinal chemistry, 87. pp. 79-88.

Ferrins, Lori and Gazdik, Michelle and Rahmani, Raphaël and Varghese, Swapna and Sykes, Melissa L. and Jones, Amy J. and Avery, Vicky M. and White, Karen L. and Ryan, Eileen and Charman, Susan A. and Kaiser, Marcel and Bergström, Christel A. S. and Baell, Jonathan B.. (2014) Pyridyl benzamides as a novel class of potent inhibitors for the kinetoplastid Trypanosoma brucei. Journal of medicinal chemistry, 57 (15). pp. 6393-6402.

Wang, Ning and Wicht, Kathryn J. and Imai, Kento and Wang, Ming-Qi and Anh Ngoc, Tran and Kiguchi, Ryo and Kaiser, Marcel and Egan, Timothy J. and Inokuchi, Tsutomu. (2014) Synthesis, β-haematin inhibition, and in vitro antimalarial testing of isocryptolepine analogues : SAR study of indolo[3,2-c]quinolines with various substituents at C2, C6, and N11. Bioorganic & medicinal chemistry, 22 (9). pp. 2629-2642.

Belluti, Federica and Uliassi, Elisa and Veronesi, Giacomo and Bergamini, Christian and Kaiser, Marcel and Brun, Reto and Viola, Angelo and Fato, Romana and Michels, Paul A. M. and Krauth-Siegel, R. Luise and Cavalli, Andrea and Bolognesi, Maria Laura. (2014) Toward the development of dual-targeted glyceraldehyde-3-phosphate dehydrogenase/trypanothione reductase inhibitors against Trypanosoma brucei and Trypanosoma cruzi. ChemMedChem : chemistry enabling drug discovery, Vol. 9, H. 2. pp. 371-382.

Reimer, Daniela and Nollmann, Friederike I. and Schultz, Katharina and Kaiser, Marcel and Bode, Helge B.. (2014) Xenortide biosynthesis by entomopathogenic xenorhabdus nematophila. Journal of natural products, 77 (8). pp. 1976-1980.

2013

Ferrins, Lori and Rahmani, Raphaël and Sykes, Melissa L. and Jones, Amy J. and Avery, Vicky M. and Teston, Eliott and Almohaywi, Basmah and Yin, Jiexiang and Smith, Jason and Hyland, Chris and White, Karen L. and Ryan, Eileen and Campbell, Michael and Charman, Susan A. and Kaiser, Marcel and Baell, Jonathan B.. (2013) 3-(Oxazolo[4,5-b]pyridin-2-yl)anilides as a novel class of potent inhibitors for the kinetoplastid Trypanosoma brucei, the causative agent for human African trypanosomiasis. European journal of medicinal chemistry, 66. pp. 450-465.

Endeshaw, Molla and Zhu, Xiaohua and He, Shanshan and Pandharkar, Trupti and Cason, Emily and Mahasenan, Kiran V. and Agarwal, Hitesh and Li, Chenglong and Munde, Manoj and Wilson, W. David and Bahar, Mark and Doskotch, Raymond W. and Kinghorn, A. Douglas and Kaiser, Marcel and Brun, Reto and Drew, Mark E. and Werbovetz, Karl A.. (2013) 8,8-dialkyldihydroberberines with potent antiprotozoal activity. Journal of natural products, Vol. 76, H. 3. pp. 311-315.

Hata, Yoshie and Raith, Melanie and Ebrahimi, Samad Nejad and Zimmermann, Stefanie and Mokoka, Tsholofelo and Naidoo, Dashnie and Fouche, Gerda and Maharaj, Vinesh and Kaiser, Marcel and Brun, Reto and Hamburger, Matthias. (2013) Antiprotozoal Isoflavan Quinones from Abrus precatorius ssp. africanus. Planta Medica, 79 (6). pp. 492-498.

Faist, Johanna and Seebacher, Werner and Kaiser, Marcel and Brun, Reto and Saf, Robert and Weis, Robert. (2013) Antiprotozoal activity of bicyclic diamines with a N-methylpiperazinyl group at the bridgehead atom. Bioorganic & medicinal chemistry : a Tetrahedron publication for the rapid dissemenination of full original research papers and critical reviews on biomolecular chemistry, medicinal chemistry and related disciplines, 21 (17). pp. 4988-4996.

Farimani, Mahdi Moridi and Ebrahimi, Samad Nejad and Salehi, Peyman and Bahadori, Mir Babak and Sonboli, Ali and Khavasi, Hamid Reza and Zimmermann, Stefanie and Kaiser, Marcel and Hamburger, Matthias. (2013) Antitrypanosomal Triterpenoid with an ε-Lactone E-Ring from Salvia urmiensis. Journal of natural products, 76 (9). pp. 1806-1809.

Graf, Fabrice E. and Ludin, Philipp and Wenzler, Tanja and Kaiser, Marcel and Brun, Reto and Pyana, Patient Pati and Büscher, Philippe and de Koning, Harry P. and Horn, David and Mäser, Pascal. (2013) Aquaporin 2 mutations in Trypanosoma brucei gambiense field isolates correlate with decreased susceptibility to pentamidine and melarsoprol. PLoS neglected tropical diseases, Vol. 7, H. 10 , e2475.

Spavieri, Jasmine and Allmendinger, Andrea and Kaiser, Marcel and Itoe, Maurice Ayamba and Blunden, Gerald and Mota, Maria M. and Tasdemir, Deniz. (2013) Assessment of dual life stage antiplasmodial activity of british seaweeds. Marine drugs, Vol. 11, H. 10. pp. 4019-4034.

Zimmermann, Stefanie and Oufir, Mouhssin and Leroux, Alejandro and Krauth-Siegel, R. Luise and Becker, Katja and Kaiser, Marcel and Brun, Reto and Hamburger, Matthias and Adams, Michael. (2013) Cynaropicrin targets the trypanothione redox system in Trypanosoma brucei. Bioorganic & medicinal chemistry, 21 (22). pp. 7202-7209.

Patra, Malay and Joshi, Tanmaya and Pierroz, Vanessa and Ingram, Katrin and Kaiser, Marcel and Ferrari, Stefano and Spingler, Bernhard and Keiser, Jennifer and Gasser, Gilles. (2013) DMSO-mediated ligand dissociation : renaissance for biological activity of N-heterocyclic-[Ru(η(6) -arene)Cl2 ] drug candidates. Chemistry : a European journal, Vol. 19, H. 44. pp. 14768-14772.

Hossain, Md Imran and Switalska, Marta and Peng, Wei and Takashima, Mariko and Wang, Ning and Kaiser, Marcel and Wietrzyk, Joanna and Dan, Shingo and Yamori, Takao and Inokuchi, Tsutomu. (2013) Design, synthesis, and in vitro cancer cell growth inhibition evaluation and antimalarial testing of trioxanes installed in cyclic 2-enoate substructures. European journal of medicinal chemistry, 69. pp. 294-309.

Lam, Cary F. C. and Pearce, A. Norrie and Tan, Shen H. and Kaiser, Marcel and Copp, Brent R.. (2013) Discovery and evaluation of thiazinoquinones as anti-protozoal agents. Marine drugs, Vol. 11, H. 9. pp. 3472-3499.

Gallé, Jean-Baptiste and Attioua, Barthélémy and Kaiser, Marcel and Rusig, Anne-Marie and Lobstein, Annelise and Vonthron-Sénécheau, Catherine. (2013) Eleganolone, a diterpene from the french marine alga Bifurcaria bifurcata inhibits growth of the human pathogens Trypanosoma brucei and Plasmodium falciparum. Marine drugs, Vol. 11, H. 3. pp. 599-610.

Hampton, Shahienaz E. and Schipani, Alessandro and Bosch-Navarrete, Cristina and Recio, Eliseo and Kaiser, Marcel and Kahnberg, Pia and González-Pacanowska, Dolores and Johansson, Nils Gunnar and Gilbert, Ian H.. (2013) Investigation of acyclic uridine amide and 5'-amido nucleoside analogues as potential inhibitors of the Plasmodium falciparum dUTPase. Bioorganic & medicinal chemistry, 21 (18). pp. 5876-5885.

Chianese, Giuseppina and Scala, Fernando and Calcinai, Barbara and Cerrano, Carlo and Dien, Henny A. and Kaiser, Marcel and Tasdemir, Deniz and Taglialatela-Scafati, Orazio. (2013) Natural and semisynthetic analogues of manadoperoxide B reveal new structural requirements for trypanocidal activity. Marine drugs, Vol. 11, H. 9. pp. 3297-3308.

Papadopoulou, Maria V. and Bloomer, William D. and Rosenzweig, Howard S. and Ashworth, Rachel and Wilkinson, Shane R. and Kaiser, Marcel and Andriani, Grasiella and Rodriguez, Ana. (2013) Novel 3-nitro-1H-1,2,4-triazole-based compounds as potential anti-Chagasic drugs : in vivo studies. Future medicinal chemistry, Vol. 5, H. 15. pp. 1763-1776.

Papadopoulou, Maria V. and Bloomer, William D. and Rosenzweig, Howard S. and Kaiser, Marcel and Chatelain, Eric and Ioset, Jean-Robert. (2013) Novel 3-nitro-1H-1,2,4-triazole-based piperazines and 2-amino-1,3-benzothiazoles as antichagasic agents. Bioorganic & medicinal chemistry, 21 (21). pp. 6600-6607.

Hwang, Jong Yeon and Smithson, David C. and Holbrook, Gloria and Zhu, Fangyi and Connelly, Michele C. and Kaiser, Marcel and Brun, Reto and Kiplin Guy, R.. (2013) Optimization of the electrophile of chloronitrobenzamide leads active against Trypanosoma brucei. Bioorganic & medicinal chemistry letters : a Tetrahedron publication for the rapid dissemination of preliminary communications on all aspects of bioorganic chemistry, medicinal chemistry, bioinorganic chemistry and related disciplines, Vol. 23, H. 14. pp. 4127-4131.

Ehmke, Veronika and Winkler, Edwin and Banner, David W. and Haap, Wolfgang and Schweizer, W. Bernd and Rottmann, Matthias and Kaiser, Marcel and Freymond, Céline and Schirmeister, Tanja and Diederich, François. (2013) Optimization of triazine nitriles as rhodesain inhibitors : structure-activity relationships, bioisosteric imidazopyridine nitriles, and X-ray crystal structure analysis with human cathepsin L. ChemMedChem : chemistry enabling drug discovery, Vol. 8, H. 6. pp. 967-975.

Reimer, Daniela and Cowles, Kimberly N. and Proschak, Anna and Nollmann, Friederike I. and Dowling, Andrea J. and Kaiser, Marcel and Constant, Richard Ffrench- and Goodrich-Blair, Heidi and Bode, Helge B.. (2013) Rhabdopeptides as insect-specific virulence factors from entomopathogenic bacteria. ChemBioChem : a European journal of chemical biology, Vol. 14, H. 15. pp. 1991-1997.

Zhou, Qiuqin and Grundmann, Florian and Kaiser, Marcel and Schiell, Matthias and Gaudriault, Sophie and Batzer, Andreas and Kurz, Michael and Bode, Helge B.. (2013) Structure and biosynthesis of xenoamicins from entomopathogenic xenorhabdus. Chemistry : a European journal, Vol. 19, H. 49. pp. 16772-16779.

Murugesan, Dinakaran and Kaiser, Marcel and White, Karen L. and Norval, Suzanne and Riley, Jennifer and Wyatt, Paul G. and Charman, Susan A. and Read, Kevin D. and Yeates, Clive and Gilbert, Ian H.. (2013) Structure-activity relationship studies of pyrrolone antimalarial agents. ChemMedChem : chemistry enabling drug discovery, Vol. 8, H. 9. pp. 1537-1544.

Lu, Wen-Jie and Wicht, Kathryn J. and Wang, Li and Imai, Kento and Mei, Zhen-Wu and Kaiser, Marcel and El Sayed, Ibrahim El Tantawy and Egan, Timothy J. and Inokuchi, Tsutomu. (2013) Synthesis and antimalarial testing of neocryptolepine analogues : addition of ester function in SAR study of 2,11-disubstituted indolo[2,3-b]quinolines. European journal of medicinal chemistry, 64. pp. 498-511.

Mei, Zhen-Wu and Wang, Li and Lu, Wen-Jie and Pang, Cui-Qing and Maeda, Tsukasa and Peng, Wei and Kaiser, Marcel and El Sayed, Ibrahim and Inokuchi, Tsutomu. (2013) Synthesis and in vitro antimalarial testing of neocryptolepines : SAR study for improved activity by introduction and modifications of side chains at C2 and C11 on indolo[2,3-b]quinolines. Journal of medicinal chemistry, 56 (4). pp. 1431-1442.

Liew, Lydia P. P. and Pearce, A. Norrie and Kaiser, Marcel and Copp, Brent R.. (2013) Synthesis and in vitro and in vivo evaluation of antimalarial polyamines. European journal of medicinal chemistry, 69. pp. 22-31.

2012

Nollmann, Friederike I. and Dowling, Andrea and Kaiser, Marcel and Deckmann, Klaus and Grösch, Sabine and Ffrench-Constant, Richard and Bode, Helge B.. (2012) Synthesis of szentiamide, a depsipeptide from entomopathogenic Xenorhabdus szentirmaii with activity against Plasmodium falciparum. Beilstein journal of organic chemistry, Vol. 8. pp. 528-533.

2011

Ślusarczyk, Sylwester and Zimmermann, Stefanie and Kaiser, Marcel and Matkowski, Adam and Hamburger, Matthias and Adams, Michael. (2011) Antiplasmodial and Antitrypanosomal Activity of Tanshinone-Type Diterpenoids from Salvia miltiorrhiza. Planta Medica, 77 (14). pp. 1594-1596.

Julianti, Tasqiah and Hata Uribe, Yoshie and Zimmermann, Stefanie and Kaiser, Marcel and Hamburger, Matthias and Adams, Michael. (2011) Antitrypanosomal sesquiterpene lactones from Saussurea costus. Fitoterapia, 82 (7). pp. 955-959.

Mokoka, Tsholofelo A. and Zimmermann, Stefanie and Julianti, Tasqiah and Hata, Yoshie and Moodley, Nivan and Cal, Monica and Adams, Michael and Kaiser, Marcel and Brun, Reto and Koorbanally, Neil and Hamburger, Matthias. (2011) In vitro screening of traditional South African malaria remedies against Trypanosoma brucei rhodesiense, Trypanosoma cruzi, Leishmania donovani, and Plasmodium falciparum. Planta Medica, 77 (14). pp. 1663-1667.

Adams, Michael and Gschwind, Sofia and Zimmermann, Stefanie and Kaiser, Marcel and Hamburger, Matthias. (2011) Renaissance remedies : antiplasmodial protostane triterpenoids from Alisma plantago-aquatica L. (Alismataceae). Journal of Ethnopharmacology, 135 (1). pp. 43-47.

2010

Orhan, Ilkay and Sener, Bilge and Kaiser, Marcel and Brun, Reto and Tasdemir, Deniz. (2010) Inhibitory activity of marine sponge-derived natural products against parasitic protozoa. Marine drugs, Vol. 8, H. 1. pp. 47-58.

Link, Andreas and Heidler, Philipp and Kaiser, Marcel and Brun, Reto. (2010) Parallel synthesis of a series of non-functional ATP/NAD analogs with activity against trypanosomatid parasites. Molecular Diversity, 14 (2). pp. 215-224.

2009

Adams, Michael and Zimmermann, Stefanie and Kaiser, Marcel and Brun, Reto and Hamburger, Matthias. (2009) A protocol for HPLC-based activity profiling for natural products with activities against tropical parasites. Natural Product Communications, 4 (10). pp. 1377-1381.

This list was generated on Thu Mar 28 17:22:52 2024 CET.