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Items where Author is "Tidwell, Richard R."

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Number of items: 10.

2017

Gillingwater, Kirsten and Kunz, Christina and Braghiroli, Christiane and Boykin, David W. and Tidwell, Richard R. and Brun, Reto. (2017) In vitro, ex vivo and in vivo activity of diamidines against Trypanosoma congolense and Trypanosoma vivax. Antimicrobial agents and chemotherapy, 61 (5). e02356-16.

2016

Pohlig, Gabriele and Bernhard, Sonja C. and Blum, Johannes and Burri, Christian and Mpanya, Alain and Lubaki, Jean-Pierre Fina and Mpoto, Alfred Mpoo and Munungu, Blaise Fungula and N'tombe, Patrick Mangoni and Deo, Gratias Kambau Manesa and Mutantu, Pierre Nsele and Kuikumbi, Florent Mbo and Mintwo, Alain Fukinsia and Munungi, Augustin Kayeye and Dala, Amadeu and Macharia, Stephen and Bilenge, Constantin Miaka Mia and Mesu, Victor Kande Betu Ku and Franco, Jose Ramon and Dituvanga, Ndinga Dieyi and Tidwell, Richard R. and Olson, Carol A.. (2016) Efficacy and safety of pafuramidine versus pentamidine maleate for treatment of first stage sleeping sickness in a randomized, comparator-controlled, international phase 3 clinical trial. PLoS neglected tropical diseases, 10 (2). e0004363.

Burri, Christian and Yeramian, Patrick D. and Allen, James L. and Merolle, Ada and Serge, Kazadi Kyanza and Mpanya, Alain and Lutumba, Pascal and Mesu, Victor Kande Betu Ku and Bilenge, Constantin Miaka Mia and Lubaki, Jean-Pierre Fina and Mpoto, Alfred Mpoo and Thompson, Mark and Munungu, Blaise Fungula and Manuel, Francisco and Josenando, Théophilo and Bernhard, Sonja C. and Olson, Carol A. and Blum, Johannes and Tidwell, Richard R. and Pohlig, Gabriele. (2016) Efficacy, safety, and dose of Pafuramidine, a new oral drug for treatment of first stage sleeping sickness, in a phase 2a clinical study and phase 2b randomized clinical studies. PLoS neglected tropical diseases, 10 (2). e0004362.

Patrick, Donald A. and Wenzler, Tanja and Yang, Sihyung and Weiser, Patrick T. and Wang, Michael Zhuo and Brun, Reto and Tidwell, Richard R.. (2016) Synthesis of novel amide and urea derivatives of thiazol-2-ethylamines and their activity against Trypanosoma brucei rhodesiense. Bioorganic & medicinal chemistry, 24 (11). pp. 2451-2465.

2015

Thuita, John K. and Wolf, Kristina K. and Murilla, Grace A. and Bridges, Arlene S. and Boykin, David W. and Mutuku, James N. and Liu, Qiang and Jones, Susan K. and Gem, Charles O. and Ching, Shelley and Tidwell, Richard R. and Wang, Michael Z. and Paine, Mary F. and Brun, Reto. (2015) Chemotherapy of second stage human African trypanosomiasis : comparison between the parenteral diamidine DB829 and its oral prodrug DB868 in vervet monkeys. PLoS neglected tropical diseases, Vol. 9, H. 2 , e3409.

2014

Patrick, Donald A. and Bakunov, Stanislav A. and Bakunova, Svetlana M. and Wenzler, Tanja and Brun, Reto and Tidwell, Richard R.. (2014) Antiprotozoal activity of dicationic 3,5-diphenylisoxazoles, their prodrugs and aza-analogues. Bioorganic & medicinal chemistry, 22 (1). pp. 559-576.

Wenzler, Tanja and Yang, Sihyung and Patrick, Donald A. and Braissant, Olivier and Ismail, Mohamed A. and Tidwell, Richard R. and Boykin, David W. and Wang, Michael Zhuo and Brun, Reto. (2014) In vitro and In vivo evaluation of 28DAP010, a novel diamidine for treatment of second-stage African sleeping sickness. Antimicrobial agents and chemotherapy, Vol. 58, H. 8. pp. 4452-4463.

2013

Thuita, John K. and Wolf, Kristina K. and Murilla, Grace A. and Liu, Qiang and Mutuku, James N. and Chen, Yao and Bridges, Arlene S. and Mdachi, Raymond E. and Ismail, Mohamed A. and Ching, Shelley and Boykin, David W. and Hall, James Edwin and Tidwell, Richard R. and Paine, Mary F. and Brun, Reto and Wang, Michael Zhuo. (2013) Safety, pharmacokinetic, and efficacy studies of oral DB868 in a first stage vervet monkey model of human African trypanosomiasis. PLoS neglected tropical diseases, Vol. 7, H. 6 , e2230.

Patrick, Donald A. and Bakunov, Stanislav A. and Bakunova, Svetlana M. and Jones, Susan Kilgore and Wenzler, Tanja and Barszcz, Todd and Kumar, Arvind and Boykin, David W. and Werbovetz, Karl A. and Brun, Reto and Tidwell, Richard R.. (2013) Synthesis and antiprotozoal activities of benzyl phenyl ether diamidine derivatives. European journal of medicinal chemistry, 67. pp. 310-324.

Patrick, Donald A. and Ismail, Mohamed A. and Arafa, Reem K. and Wenzler, Tanja and Zhu, Xiaohua and Pandharkar, Trupti and Jones, Susan Kilgore and Werbovetz, Karl A. and Brun, Reto and Boykin, David W. and Tidwell, Richard R.. (2013) Synthesis and antiprotozoal activity of dicationic m-terphenyl and 1,3-dipyridylbenzene derivatives. Journal of medicinal chemistry, 56 (13). pp. 5473-5494.

This list was generated on Thu Mar 28 17:02:32 2024 CET.