Items where Author is "Scapozza, Leonardo"

2015

Seebacher, Werner and Wolkinger, Volker and Faist, Johanna and Kaiser, Marcel and Brun, Reto and Saf, Robert and Bucar, Franz and Gröblacher, Barbara and Brantner, Adelheid and Merino, Virginia and Kalia, Yogeshvar and Scapozza, Leonardo and Perozzo, Remo and Weis, Robert. (2015) Synthesis of 3-azabicyclo[3.2.2]nonanes and their antiprotozoal activities. Bioorganic & medicinal chemistry letters, Vol. 25, H. 7. pp. 1390-1393.

2014

Wang, Tai and Bisson, William H. and Mäser, Pascal and Scapozza, Leonardo and Picard, Didier. (2014) Differences in conformational dynamics between Plasmodium falciparum and human Hsp90 orthologues enable the structure-based discovery of pathogen-selective inhibitors. Journal of medicinal chemistry, 57 (6). pp. 2524-2535.

2013

Belluti, Federica and Perozzo, Remo and Lauciello, Leonardo and Colizzi, Francesco and Kostrewa, Dirk and Bisi, Alessandra and Gobbi, Silvia and Rampa, Angela and Bolognesi, Maria Laura and Recanatini, Maurizio and Brun, Reto and Scapozza, Leonardo and Cavalli, Andrea. (2013) Design, synthesis, and biological and crystallographic evaluation of novel inhibitors of Plasmodium falciparum enoyl-ACP-reductase (PfFabI). Journal of medicinal chemistry, 56 (19). pp. 7516-7526.

Pieretti, Simone and Haanstra, Jurgen R. and Mazet, Muriel and Perozzo, Remo and Bergamini, Christian and Prati, Federica and Fato, Romana and Lenaz, Giorgio and Capranico, Giovanni and Brun, Reto and Bakker, Barbara M. and Michels, Paul A. M. and Scapozza, Leonardo and Bolognesi, Maria Laura and Cavalli, Andrea. (2013) Naphthoquinone derivatives exert their antitrypanosomal activity via a multi-target mechanism. PLoS neglected tropical diseases, Vol. 7 , e2012.