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Items where Author is "Gasser, Gilles"

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Number of items: 11.

2020

Buchter, Valentin and Ong, Yih Ching and Mouvet, François and Ladaycia, Abdallah and Lepeltier, Elise and Rothlisberger, Ursula and Keiser, Jennifer and Gasser, Gilles. (2020) Multidisciplinary preclinical investigations on three oxamniquine analogues as novel drug candidates for schistosomiasis. Chemistry (Weinheim an der Bergstrasse, Germany), 26 (66). pp. 15232-15241.

Lin, Yan and Ong, Yih Ching and Keller, Sarah and Karges, Johannes and Bouchene, Rafika and Manoury, Eric and Blacque, Olivier and Müller, Joachim and Anghel, Nicoleta and Hemphill, Andrew and Häberli, Cécile and Taki, Aya C. and Gasser, Robin B. and Cariou, Kevin and Keiser, Jennifer and Gasser, Gilles. (2020) Synthesis, characterization and antiparasitic activity of organometallic derivatives of the anthelmintic drug albendazole. Dalton Transactions, 49 (20). pp. 6616-6626.

2018

Buchter, Valentin and Hess, Jeannine and Gasser, Gilles and Keiser, Jennifer. (2018) Assessment of tegumental damage to Schistosoma mansoni and S. haematobium after in vitro exposure to ferrocenyl, ruthenocenyl and benzyl derivatives of oxamniquine using scanning electron microscopy. Parasites and Vectors, 11. p. 580.

2017

Hess, Jeannine and Panic, Gordana and Patra, Malay and Mastrobuoni, Luciano and Spingler, Bernhard and Roy, Saonli and Keiser, Jennifer and Gasser, Gilles. (2017) Ferrocenyl, ruthenocenyl, and benzyl oxamniquine derivatives with cross-species activity against Schistosoma mansoni and Schistosoma haematobium. ACS infectious diseases, 3 (9). pp. 645-652.

2016

Clède, Sylvain and Cowan, Noemi and Lambert, François and Bertrand, Hélène C. and Rubbiani, Riccardo and Patra, Malay and Hess, Jeannine and Sandt, Christophe and Trcera, Nicolas and Gasser, Gilles and Keiser, Jennifer and Policar, Clotilde. (2016) Bimodal x-ray and infrared imaging of an organometallic derivative of praziquantel in Schistosoma mansoni. ChemBioChem, 17 (11). pp. 1004-1007.

2015

Hess, Jeannine and Keiser, Jennifer and Gasser, Gilles. (2015) Toward organometallic antischistosomal drug candidates. Future medicinal chemistry, Vol. 7, H. 6. pp. 821-830.

2014

Meister, Isabel and Ingram-Sieber, Katrin and Cowan, Noemi and Todd, Matthew and Robertson, Murray N. and Meli, Claudia and Patra, Malay and Gasser, Gilles and Keiser, Jennifer. (2014) Activity of praziquantel enantiomers and main metabolites against Schistosoma mansoni. Antimicrobial agents and chemotherapy, Vol. 58, H. 9. pp. 5466-5472.

Patra, Malay and Bauman, Andreas and Mari, Cristina and Fischer, Christiane A. and Blacque, Olivier and Häussinger, Daniel and Gasser, Gilles and Mindt, Thomas L.. (2014) An octadentate bifunctional chelating agent for the development of stable zirconium-89 based molecular imaging probes. Chemical Communications, 50 (78). pp. 11523-11525.

Keiser, Jennifer and Vargas, Mireille and Rubbiani, Riccardo and Gasser, Gilles and Biot, Christophe. (2014) In vitro and in vivo antischistosomal activity of ferroquine derivatives. Parasites and Vectors, 7 (424).

2013

Patra, Malay and Joshi, Tanmaya and Pierroz, Vanessa and Ingram, Katrin and Kaiser, Marcel and Ferrari, Stefano and Spingler, Bernhard and Keiser, Jennifer and Gasser, Gilles. (2013) DMSO-mediated ligand dissociation : renaissance for biological activity of N-heterocyclic-[Ru(η(6) -arene)Cl2 ] drug candidates. Chemistry : a European journal, Vol. 19, H. 44. pp. 14768-14772.

Patra, Malay and Ingram, Katrin and Leonidova, Anna and Pierroz, Vanessa and Ferrari, Stefano and Robertson, Murray N. and Todd, Matthew H. and Keiser, Jennifer and Gasser, Gilles. (2013) In vitro metabolic profile and in vivo antischistosomal activity studies of (η(6)-praziquantel)Cr(CO)3 derivatives. Journal of medicinal chemistry, 56 (22). pp. 9192-9198.

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