Items where Author is "Baell, Jonathan B."

2019

Le, Thuy G. and Kundu, Abhijit and Ghoshal, Atanu and Nguyen, Nghi H. and Preston, Sarah and Jiao, Yaqing and Ruan, Banfeng and Xue, Lian and Huang, Fei and Keiser, Jennifer and Hofmann, Andreas and Chang, Bill C. H. and Garcia-Bustos, Jose and Wells, Timothy N. C. and Palmer, Michael J. and Jabbar, Abdul and Gasser, Robin B. and Baell, Jonathan B.. (2019) Novel 1-methyl-1 H-pyrazole-5-carboxamide derivatives with potent anthelmintic activity. Journal of medicinal chemistry, 62 (7). pp. 3367-3380.

Le, Thuy and Kundu, Abhijit and Ghoshal, Atanu and Nguyen, Nghi and Preston, Sarah and Jiao, Yaqing and Ruan, Banfeng and Xue, Lian and Huang, Fei and Keiser, Jennifer and Hofmann, Andreas and Chang, Bill and Garcia-Bustos, Jose and Wells, Timothy N. C. and Palmer, Michael J. and Jabbar, Abdul and Gasser, Robin B. and Baell, Jonathan B.. (2019) Structure-activity relationship studies of tolfenpyrad reveal sub-nanomolar inhibitors of Haemonchus contortus development. Journal of medicinal chemistry, 62 (2). pp. 1036-1053.

2018

Le, Thuy G. and Kundu, Abhijit and Ghoshal, Atanu and Nguyen, Nghi H. and Preston, Sarah and Jiao, Yaqing and Ruan, Banfeng and Xue, Lian and Huang, Fei and Keiser, Jennifer and Hofmann, Andreas and Chang, Bill C. H. and Garcia-Bustos, Jose and Jabbar, Abdul and Wells, Timothy N. C. and Palmer, Michael J. and Gasser, Robin B. and Baell, Jonathan B.. (2018) Optimization of novel 1-methyl-1 h-pyrazole-5-carboxamides leads to high potency larval development inhibitors of the barber's pole worm. Journal of medicinal chemistry, 61 (23). pp. 10875-10894.

2017

Preston, Sarah and Jiao, Yaqing and Baell, Jonathan B. and Keiser, Jennifer and Crawford, Simon and Koehler, Anson V. and Wang, Tao and Simpson, Moana M. and Kaplan, Ray M. and Cowley, Karla J. and Simpson, Kaylene J. and Hofmann, Andreas and Jabbar, Abdul and Gasser, Robin B.. (2017) Screening of the 'Open Scaffolds' collection from Compounds Australia identifies a new chemical entity with anthelmintic activities against different developmental stages of the barber's pole worm and other parasitic nematodes. International Journal for Parasitology: Drugs and Drug Resistance, 7 (3). pp. 286-294.

2016

Russell, Stephanie and Rahmani, Raphaël and Jones, Amy J. and Newson, Harriet L. and Neilde, Kevin and Cotillo, Ignacio and Rahmani Khajouei, Marzieh and Ferrins, Lori and Qureishi, Sana and Nguyen, Nghi and Martinez-Martinez, Maria S. and Weaver, Donald F. and Kaiser, Marcel and Riley, Jennifer and Thomas, John and De Rycker, Manu and Read, Kevin D. and Flematti, Gavin R. and Ryan, Eileen and Tanghe, Scott and Rodriguez, Ana and Charman, Susan A. and Kessler, Albane and Avery, Vicky M. and Baell, Jonathan B. and Piggott, Matthew J.. (2016) Hit-to-lead optimization of a novel class of potent, broad-spectrum trypanosomacides. Journal of Medicinal Chemistry, 59 (21). pp. 9686-9720.

Williamson, Alice E. and Ylioja, Paul M. and Robertson, Murray N. and Antonova-Koch, Yevgeniya and Avery, Vicky and Baell, Jonathan B. and Batchu, Harikrishna and Batra, Sanjay and Burrows, Jeremy N. and Bhattacharyya, Soumya and Calderon, Felix and Charman, Susan A. and Clark, Julie and Crespo, Benigno and Dean, Matin and Debbert, Stefan L. and Delves, Michael and Dennis, Adelaide S. M. and Deroose, Frederik and Duffy, Sandra and Fletcher, Sabine and Giaever, Guri and Hallyburton, Irene and Gamo, Francisco-Javier and Gebbia, Marinella and Guy, R. Kiplin and Hungerford, Zoe and Kirk, Kiaran and Lafuente-Monasterio, Maria J. and Lee, Anna and Meister, Stephan and Nislow, Corey and Overington, John P. and Papadatos, George and Patiny, Luc and Pham, James and Ralph, Stuart A. and Ruecker, Andrea and Ryan, Eileen and Southan, Christopher and Srivastava, Kumkum and Swain, Chris and Tarnowski, Matthew J. and Thomson, Patrick and Turner, Peter and Wallace, Iain M. and Wells, Timothy N. C. and White, Karen and White, Laura and Willis, Paul and Winzeler, Elizabeth A. and Wittlin, Sergio and Todd, Matthew H.. (2016) Open source drug discovery : highly potent antimalarial compounds derived from the tres cantos arylpyrroles. ACS central science, 2 (10). pp. 687-701.

2015

Rahmani, Raphaël and Ban, Kung and Jones, Amy J. and Ferrins, Lori and Ganame, Danny and Sykes, Melissa L. and Avery, Vicky M. and White, Karen L. and Ryan, Eileen and Kaiser, Marcel and Charman, Susan A. and Baell, Jonathan B.. (2015) 6-Arylpyrazine-2-carboxamides : a new core for Trypanosoma brucei inhibitors. Journal of medicinal chemistry, 58 (17). pp. 6753-6765.

2014

Ferrins, Lori and Gazdik, Michelle and Rahmani, Raphaël and Varghese, Swapna and Sykes, Melissa L. and Jones, Amy J. and Avery, Vicky M. and White, Karen L. and Ryan, Eileen and Charman, Susan A. and Kaiser, Marcel and Bergström, Christel A. S. and Baell, Jonathan B.. (2014) Pyridyl benzamides as a novel class of potent inhibitors for the kinetoplastid Trypanosoma brucei. Journal of medicinal chemistry, 57 (15). pp. 6393-6402.

2013

Ferrins, Lori and Rahmani, Raphaël and Sykes, Melissa L. and Jones, Amy J. and Avery, Vicky M. and Teston, Eliott and Almohaywi, Basmah and Yin, Jiexiang and Smith, Jason and Hyland, Chris and White, Karen L. and Ryan, Eileen and Campbell, Michael and Charman, Susan A. and Kaiser, Marcel and Baell, Jonathan B.. (2013) 3-(Oxazolo[4,5-b]pyridin-2-yl)anilides as a novel class of potent inhibitors for the kinetoplastid Trypanosoma brucei, the causative agent for human African trypanosomiasis. European journal of medicinal chemistry, 66. pp. 450-465.